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PubMed code 10673095

Compile data set for download or QSAR
Found 2 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 1


(Homo sapiens (Human))
BDBM17657
PNG
((2S)-2-aminopentanedioic acid | (S)-Glu | D-Glutam...)
Show SMILES N[C@@H](CCC(O)=O)C(O)=O
Show InChI InChI=1S/C5H9NO4/c6-3(5(9)10)1-2-4(7)8/h3H,1-2,6H2,(H,7,8)(H,9,10)/t3-/m0/s1
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UniProtKB/SwissProt

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KEGG
MMDB
PC cid
PC sid
PDB
UniChem

Patents


Similars

Article
PubMed
n/an/an/an/a 1.05E+3n/an/an/an/a



CNRS

Curated by ChEMBL


Assay Description
Effect of compound on Metabotropic glutamate receptor 1 expressed in HEK 293 cells was determined by measuring IP production relative to glutamate


Bioorg Med Chem Lett 10: 129-33 (2000)


Article DOI: 10.1016/s0960-894x(99)00641-1
BindingDB Entry DOI: 10.7270/Q2P84CFG
More data for this
Ligand-Target Pair
Metabotropic glutamate receptor 1


(Homo sapiens (Human))
BDBM50084962
PNG
((2S,3S,4S)-2-Amino-3,4-dihydroxy-pentanedioic acid...)
Show SMILES N[C@@H]([C@H](O)[C@H](O)C(O)=O)C(O)=O
Show InChI InChI=1S/C5H9NO6/c6-1(4(9)10)2(7)3(8)5(11)12/h1-3,7-8H,6H2,(H,9,10)(H,11,12)/t1-,2-,3-/m0/s1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/an/an/a 2.57E+5n/an/an/an/a



CNRS

Curated by ChEMBL


Assay Description
Effect of compound on Metabotropic glutamate receptor 1 expressed in HEK 293 cells was determined by measuring IP production relative to glutamate


Bioorg Med Chem Lett 10: 129-33 (2000)


Article DOI: 10.1016/s0960-894x(99)00641-1
BindingDB Entry DOI: 10.7270/Q2P84CFG
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%