Found 48 Enz. Inhib. hit(s) with all data for entry = 50036927 
Affinity DataKi: 0.160nMAssay Description:Binding affinity against cloned human Opioid receptor delta 1 transfected onto CHO cells using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Binding affinity against Opioid receptor kappa 1 in guinea pig brain membranes using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Opioid receptor mu 1 in guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity against Opioid receptor mu 1 in guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.640nMAssay Description:Binding affinity against cloned human Opioid receptor mu 1 transfected onto CHO cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Binding affinity against cloned human opioid Opioid receptor mu 1 transfected onto CHO cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity against Opioid receptor kappa 1 in guinea pig brain membranes using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 0.840nMAssay Description:Binding affinity against cloned human opioid Opioid receptor kappa 1 transfected onto CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity against Opioid receptor mu 1 in guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity against cloned human Opioid receptor kappa 1 transfected onto CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity against Opioid receptor mu 1 in guinea pig brain membranes using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity against cloned human opioid mu receptors transfected onto CHO cells using [3H]DAMGOMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:Binding affinity against Opioid receptor kappa 1 in guinea pig brain membranes using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity against cloned human Opioid receptor kappa 1 transfected onto CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Binding affinity against cloned human Opioid receptor delta 1 transfected onto CHO cells using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Binding affinity against cloned human Opioid receptor mu 1 transfected onto CHO cells using [3H]DAMGOMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Binding affinity against Opioid receptor delta 1 in guinea pig brain membranes using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against cloned human Opioid receptor delta 1 transfected onto CHO cells using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Bristol
Curated by ChEMBL
University Of Bristol
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Binding affinity against Opioid receptor kappa 1 in guinea pig brain membranes using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity against cloned human opioid Opioid receptor kappa 1 transfected onto CHO cells using [3H]U-69593More data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against cloned human Opioid receptor delta 1 transfected onto CHO cells using [3H]Cl-DPDPEMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor mu 1 (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor mu 1 (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor mu 1 (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.800nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.610nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 161nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor mu 1 (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human opioid mu receptor transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor mu 1 (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 559nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor kappa 1 (U-69,593) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 7.30nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human opioid mu receptors (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.660nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human oOpioid receptor mu 1 (DAMGO) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human oOpioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 19nMAssay Description:EC50 for binding of [35S]- GTPdeltaS in cloned human Opioid receptor delta 1 (Cl-DPDPE) transfected onto CHO cellsMore data for this Ligand-Target Pair
