Compile Data Set for Download or QSAR
maximum 50k data
Found 90 Enz. Inhib. hit(s) with all data for entry = 50048517
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  0.269nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  1.60nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  6nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  6.5nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  10nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  10nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  11nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  31nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  34nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM82423(CAS_132947 | NSC_132947 | TRIPITRAMINE)
Affinity DataKi:  38nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81452(CAS_91533 | Dimethindene | NSC_91533)
Affinity DataKi:  45nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  66nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  93nMAssay Description:In vitro transcriptional activation in CV-1 cells expressing human Gal4-PPAR gamma ligand binding domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  107nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81452(CAS_91533 | Dimethindene | NSC_91533)
Affinity DataKi:  191nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81452(CAS_91533 | Dimethindene | NSC_91533)
Affinity DataKi:  263nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219396(CHEMBL21716)
Affinity DataKi:  324nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219395(CHEMBL278074)
Affinity DataKi:  331nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81452(CAS_91533 | Dimethindene | NSC_91533)
Affinity DataKi:  407nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219393(CHEMBL21321)
Affinity DataKi:  417nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50076089((3S,3aR,4R,4aS,8aR,9aS)-3-Methyl-4-[2-((R)-1-methy...)
Affinity DataKi:  490nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81901(AF-DX 384 | CAS_119356 | CHEMBL279453 | NSC_119356)
Affinity DataKi:  537nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM81452(CAS_91533 | Dimethindene | NSC_91533)
Affinity DataKi:  794nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219393(CHEMBL21321)
Affinity DataKi:  891nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219396(CHEMBL21716)
Affinity DataKi:  977nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219395(CHEMBL278074)
Affinity DataKi:  1.05E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219393(CHEMBL21321)
Affinity DataKi:  1.23E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219393(CHEMBL21321)
Affinity DataKi:  1.23E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M5 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219395(CHEMBL278074)
Affinity DataKi:  1.26E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219396(CHEMBL21716)
Affinity DataKi:  1.48E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219396(CHEMBL21716)
Affinity DataKi:  1.70E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219393(CHEMBL21321)
Affinity DataKi:  1.70E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219396(CHEMBL21716)
Affinity DataKi:  1.74E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219395(CHEMBL278074)
Affinity DataKi:  1.82E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219395(CHEMBL278074)
Affinity DataKi:  2.09E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219394(CHEMBL20732)
Affinity DataKi:  7.08E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219391(CHEMBL280684)
Affinity DataKi:  7.41E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219350(CHEMBL279225)
Affinity DataKi:  9.12E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219354(CHEMBL21509)
Affinity DataKi:  9.55E+3nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219391(CHEMBL280684)
Affinity DataKi:  1.00E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219392(CHEMBL278129)
Affinity DataKi:  1.05E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219391(CHEMBL280684)
Affinity DataKi:  1.15E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219392(CHEMBL278129)
Affinity DataKi:  1.20E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M1 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219394(CHEMBL20732)
Affinity DataKi:  1.20E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219354(CHEMBL21509)
Affinity DataKi:  1.20E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219394(CHEMBL20732)
Affinity DataKi:  1.23E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219391(CHEMBL280684)
Affinity DataKi:  1.26E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M4 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219354(CHEMBL21509)
Affinity DataKi:  1.26E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219394(CHEMBL20732)
Affinity DataKi:  1.41E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M3 expressed in CHO cells by [3H]-NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
University Of Mainz

Curated by ChEMBL
LigandPNGBDBM50219349(CHEMBL21328)
Affinity DataKi:  1.41E+4nMAssay Description:Affinity for Muscarinic acetylcholine receptor M2 expressed in CHO cells by [3H]NMS displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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