TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 1.75E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.86E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 3.87E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Osaka University Of Pharmaceutical Sciences
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair