Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50011686
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109332(1-[4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyr...)
Affinity DataIC50:  120nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109338(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-py...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109319(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50:  220nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109316(1-[4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyr...)
Affinity DataIC50:  240nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109337(1-[5-Butyl-4-(4-fluoro-phenyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109339(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-py...)
Affinity DataIC50:  300nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109329(CHEMBL143664 | [4-(4-Fluoro-phenyl)-5-hexyl-2,6-di...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109323(CHEMBL140514 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  400nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331(CHEMBL24616 | [4-(4-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109341(CHEMBL140268 | [4-(4-Fluoro-phenyl)-5-heptyl-2,6-d...)
Affinity DataIC50:  700nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109318(CHEMBL143698 | [5-Butyl-4-(4-fluoro-phenyl)-2,6-di...)
Affinity DataIC50:  750nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109325(CHEMBL140586 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109327(CHEMBL143609 | [5-Ethyl-4-(4-fluoro-phenyl)-2,6-di...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109336((2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-m...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109317((5-Ethyl-2,6-diisopropyl-4-phenyl-pyridin-3-yl)-me...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109315(CHEMBL140636 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322(CHEMBL114761 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibitory concentration of the compound against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109330(CHEMBL140209 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322(CHEMBL114761 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109321(CHEMBL140267 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109320(CHEMBL436011 | [4-(4-Fluoro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109324(4-(4-Fluoro-phenyl)-5-hydroxymethyl-2,6-diisopropy...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109334((2,6-Diethyl-5-pentyl-4-phenyl-pyridin-3-yl)-metha...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109333(CHEMBL346859 | [4-(4-Fluoro-phenyl)-5-hydroxymethy...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109335((2,5,6-Triethyl-4-phenyl-pyridin-3-yl)-methanol | ...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109328((2,6-Dimethyl-5-pentyl-4-phenyl-pyridin-3-yl)-meth...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109340((5-Ethyl-2,6-dimethyl-4-phenyl-pyridin-3-yl)-metha...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed