Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50011782
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50026486((Z)-7-Phenyl-7-pyridin-3-yl-hept-6-enoic acid | 7-...)
Affinity DataIC50:  0.900nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110458(5-(Phenyl-pyridin-3-yl-methyleneaminooxy)-pentanoi...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110447(CHEMBL352120 | ethyl 5-{[1-(3-{4-[6-(2-chloropheny...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110446(5-{[1-{3-[6-(2-chlorophenyl)-1,4-dimethyl-7,8,9,10...)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110456(5-([3-{1-[6-(2-chlorophenyl)-1,4-dimethyl-7,8,9,10...)
Affinity DataIC50:  41nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110457(CHEMBL349982 | ethyl 5-{[1-(4-{2-[6-(2-chloropheny...)
Affinity DataIC50:  58nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110452(5-[(3-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  59nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109127(5-[(3-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  65nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110443(CHEMBL423993 | ethyl 5-{[1-{3-[6-(2-chlorophenyl)-...)
Affinity DataIC50:  65nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110450(6-(2-Chlorophenyl)-3-[3-[(E/Z)-6-ethoxycarbonyl-1-...)
Affinity DataIC50:  68nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110449(5-[(4-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  69nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50109129(5-[(4-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110455(6-(2-Chlorophenyl)-3-[4-[(E/Z)-6-ethoxycarbonyl-1-...)
Affinity DataIC50:  72nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110451(5-[(4-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50:  80nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110453(2-(1,4-oxazinan-4-yl)ethyl 5-{[1-{3-[6-(2-chloroph...)
Affinity DataIC50:  151nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110444(CHEMBL351562 | benzyl 5-{[1-{3-[6-(2-chlorophenyl)...)
Affinity DataIC50:  465nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110442(1N-propyl-5-{[1-{3-[6-(2-chlorophenyl)-1,4-dimethy...)
Affinity DataIC50:  540nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110454(5-[(2-[1,4-dimethyl-6-(2-chloro-phenyl)-7,8,9,10-t...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110445(2-(1,4-dimethyl-7,8,9,10-tetrahydro-4H-pyrido[4',3...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Nikken Chemicals

Curated by ChEMBL
LigandPNGBDBM50110448(3-(3-pyridyl)propyl 5-{[1-{3-[6-(2-chlorophenyl)-1...)
Affinity DataIC50: >1.00E+3nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed