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Found 21 Enz. Inhib. hit(s) with all data for entry = 50011803
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50084617(((7-carbamimidoyl-naphthalen-2-ylmethyl)-{4-[1-(1-...)
Affinity DataKi:  2.30nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50097771(3-[(Z)-AMINO(IMINO)METHYL]-N-[2-(4-BENZOYL-1-PIPER...)
Affinity DataKi:  16nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110746(3-Carbamimidoyl-N-{2-[4-(4-chloro-phenyl)-piperazi...)
Affinity DataKi:  16nMAssay Description:Inhibitory concentration against human Coagulation factor Xa(fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110748((3-Carbamimidoyl-benzoylamino)-phenyl-acetic acid ...)
Affinity DataKi:  26nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110745(3-(6-Carbamimidoyl-naphthalen-2-yl)-2-{4-[1-(1-imi...)
Affinity DataKi:  41nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50084617(((7-carbamimidoyl-naphthalen-2-ylmethyl)-{4-[1-(1-...)
Affinity DataKi:  159nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50038002(Benzamidine (Protonated) | CHEMBL20936 | CHEMBL537...)
Affinity DataKi:  200nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110749(CHEMBL417827 | N-{[(4-Aminomethyl-cyclohexylmethyl...)
Affinity DataKi:  220nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110745(3-(6-Carbamimidoyl-naphthalen-2-yl)-2-{4-[1-(1-imi...)
Affinity DataKi:  630nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50097771(3-[(Z)-AMINO(IMINO)METHYL]-N-[2-(4-BENZOYL-1-PIPER...)
Affinity DataKi:  980nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110746(3-Carbamimidoyl-N-{2-[4-(4-chloro-phenyl)-piperazi...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory concentration against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110748((3-Carbamimidoyl-benzoylamino)-phenyl-acetic acid ...)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110746(3-Carbamimidoyl-N-{2-[4-(4-chloro-phenyl)-piperazi...)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110745(3-(6-Carbamimidoyl-naphthalen-2-yl)-2-{4-[1-(1-imi...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibitory concentration against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110747(2-(3-Carbamimidoyl-benzoylamino)-3-naphthalen-2-yl...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibitory concentration against human Coagulation factor Xa (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110749(CHEMBL417827 | N-{[(4-Aminomethyl-cyclohexylmethyl...)
Affinity DataKi:  7.40E+3nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110748((3-Carbamimidoyl-benzoylamino)-phenyl-acetic acid ...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibitory concentration against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50084617(((7-carbamimidoyl-naphthalen-2-ylmethyl)-{4-[1-(1-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory concentration against thrombin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50110747(2-(3-Carbamimidoyl-benzoylamino)-3-naphthalen-2-yl...)
Affinity DataKi:  1.25E+4nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50097774(CHEMBL20912 | N-{[(4-Aminomethyl-cyclohexylmethyl)...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Bos taurus (bovine))
Protherics Molecular Design

Curated by ChEMBL
LigandPNGBDBM50038002(Benzamidine (Protonated) | CHEMBL20936 | CHEMBL537...)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibitory concentration against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed