Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50011828
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50111008(5-{3-[4-(5-Methyl-2-phenyl-thiazol-4-ylmethoxy)-ph...)
Affinity DataEC50:  813nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50049240((+-)-5-((4-(2-(5-ethyl-2-pyridinyl)ethoxy)phenyl)m...)
Affinity DataEC50:  490nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alpha; values in the parentheses indicates 95% confidence intervalMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50111006(5-{3-[4-(2-Furan-2-yl-5-methyl-oxazol-4-ylmethoxy)...)
Affinity DataEC50:  8.87nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50111010(5-{3-[4-(5-Methyl-2-naphthalen-2-yl-oxazol-4-ylmet...)
Affinity DataEC50:  29.3nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50111008(5-{3-[4-(5-Methyl-2-phenyl-thiazol-4-ylmethoxy)-ph...)
Affinity DataEC50:  269nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50111009(5-{3-[4-(5-Methyl-2-phenyl-oxazol-4-ylmethoxy)-phe...)
Affinity DataEC50:  119nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma/Retinoic acid receptor RXR-alpha(Homo sapiens (Human))
Takeda Chemical Industries

Curated by ChEMBL
LigandPNGBDBM50111007(5-{3-[6-(5-Methyl-2-phenyl-oxazol-4-ylmethoxy)-pyr...)
Affinity DataEC50:  16.5nMAssay Description:Transcriptional activation in COS cells expressing PPAR gamma and RXR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed