Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50035250
TargetThymidylate kinase(Mycobacterium tuberculosis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118628((R)-1-((R)-4-Azido-5-methylphosphate-tetrahydro-fu...)
Affinity DataKi:  1.00E+4nMAssay Description:Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118625((R)-1-((R)-3-Chloro-4-hydroxy-5-methylphosphate-te...)
Affinity DataKi:  1.90E+4nMAssay Description:Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118627((R)-1-((R)-4-Amino-3-hydroxy-5-methylphosphate-tet...)
Affinity DataKi:  2.70E+4nMAssay Description:Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118623((R)-1-((R)-3-Fluoro-4-hydroxy-5-methylphosphate-te...)
Affinity DataKi:  4.30E+4nMAssay Description:Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118624((R)-1-((R)-3-Amino-4-hydroxy-5-methylphosphate-tet...)
Affinity DataKi:  5.50E+4nMAssay Description:Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate kinase(Mycobacterium tuberculosis)
Ghent University

Curated by ChEMBL
LigandPNGBDBM50118626((R)-1-((R)-4-Amino-5-methylphosphate-tetrahydro-fu...)
Affinity DataKi:  2.35E+5nMAssay Description:Compound was tested for binding affinity against Mycobacterium tuberculosis thymidine monophosphate kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed