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Found 45 Enz. Inhib. hit(s) with all data for entry = 50042174
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50220136(3-[2-{1-[3,5-di(trifluoromethyl)phenyl]ethoxy}-3-(...)
Affinity DataIC50:  0.100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421571(CHEMBL111303)
Affinity DataIC50:  0.794nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421552(CHEMBL108200)
Affinity DataIC50:  1nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421563(CHEMBL111176)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421561(CHEMBL419742)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421562(CHEMBL108889)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421564(CHEMBL107941)
Affinity DataIC50:  2.5nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421560(CHEMBL108667)
Affinity DataIC50:  3.20nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421554(CHEMBL107875)
Affinity DataIC50:  3.20nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421564(CHEMBL107941)
Affinity DataIC50:  3.20nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421573(CHEMBL321892)
Affinity DataIC50:  5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421556(CHEMBL109183)
Affinity DataIC50:  5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421567(CHEMBL109937)
Affinity DataIC50:  5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421558(CHEMBL432627)
Affinity DataIC50:  6.30nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421568(CHEMBL108422)
Affinity DataIC50:  6.30nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM30130(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)
Affinity DataIC50:  6.30nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421558(CHEMBL432627)
Affinity DataIC50:  7.90nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421555(CHEMBL111244)
Affinity DataIC50:  7.90nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421560(CHEMBL108667)
Affinity DataIC50:  10nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421553(CHEMBL320535)
Affinity DataIC50:  13nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421566(CHEMBL107829)
Affinity DataIC50:  13nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421565(CHEMBL107831)
Affinity DataIC50:  13nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421553(CHEMBL320535)
Affinity DataIC50:  16nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421563(CHEMBL111176)
Affinity DataIC50:  25nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421565(CHEMBL107831)
Affinity DataIC50:  25nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421569(CHEMBL108822)
Affinity DataIC50:  25nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421566(CHEMBL107829)
Affinity DataIC50:  32nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421572(CHEMBL110086)
Affinity DataIC50:  40nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421570(CHEMBL320544)
Affinity DataIC50:  50nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421559(CHEMBL109514)
Affinity DataIC50:  100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421570(CHEMBL320544)
Affinity DataIC50:  100nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421557(CHEMBL111304)
Affinity DataIC50:  100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421559(CHEMBL109514)
Affinity DataIC50:  158nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421562(CHEMBL108889)
Affinity DataIC50:  200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421556(CHEMBL109183)
Affinity DataIC50:  200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421573(CHEMBL321892)
Affinity DataIC50:  200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421552(CHEMBL108200)
Affinity DataIC50:  200nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421571(CHEMBL111303)
Affinity DataIC50:  200nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421568(CHEMBL108422)
Affinity DataIC50:  251nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421567(CHEMBL109937)
Affinity DataIC50:  251nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421561(CHEMBL419742)
Affinity DataIC50:  251nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421572(CHEMBL110086)
Affinity DataIC50:  316nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421554(CHEMBL107875)
Affinity DataIC50:  316nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421555(CHEMBL111244)
Affinity DataIC50:  398nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells using [3H]-substance P as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50421557(CHEMBL111304)
Affinity DataIC50:  1.00E+3nMAssay Description:Binding affinity against Serotonin transporter in rat cerebral cortex using [3H]paroxetine binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed