Affinity DataKi: 0.0620nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 0.810nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.880nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80 (Opioid receptor delta 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by SNC80More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Opioid receptor delta 1 binding affinity was determined by inhibition of binding of [3H]DADLE to rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by DAMGO (Opioid receptor mu 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:The ability of compound to inhibit [35S]GTP-delta-S binding in guinea pig caudate stimulated by U69,593 (Opioid receptor kappa 1) antagonistMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 94nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 106nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 115nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 134nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 149nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 151nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 171nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 185nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 233nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 238nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 349nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 370nMAssay Description:Binding affinity at delta opioid receptor 1 in rat brain membrane by [3H]DADLE displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 378nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 395nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair
Affinity DataKi: 409nMAssay Description:Binding affinity at mu opioid receptor 1 in rat brain membrane by [3H]DAMGO displacement.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Innsbruck
Curated by ChEMBL
University Of Innsbruck
Curated by ChEMBL
Affinity DataKi: 504nMAssay Description:Binding affinity at kappa opioid receptor 1 in guinea pig brain by [3H]U-69593 displacement.More data for this Ligand-Target Pair