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Found 33 Enz. Inhib. hit(s) with all data for entry = 50012865
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123521(CHEMBL317791 | [2'-(2-Pyridin-2-yl-ethylcarbamoyl)...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123507(2'-[(3-Phenyl-butyrylamino)-methyl]-biphenyl-2-car...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123525(CHEMBL146482 | [2'-(1-Carbamoyl-3-methyl-butylcarb...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123528(CHEMBL148356 | {2-[2-(Cyclopropylmethyl-carbamoyl)...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123521(CHEMBL317791 | [2'-(2-Pyridin-2-yl-ethylcarbamoyl)...)
Affinity DataIC50:  500nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.3 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123511(CHEMBL148210 | [6,6'-Dimethyl-2'-(2-pyridin-2-yl-e...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123508(CHEMBL148159 | [2'-(2-Pyridin-2-yl-ethylcarbamoyl)...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123511(CHEMBL148210 | [6,6'-Dimethyl-2'-(2-pyridin-2-yl-e...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123518(CHEMBL147381 | [2'-(3-Methyl-butylcarbamoyl)-biphe...)
Affinity DataIC50:  800nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123529(CHEMBL147039 | [6,6'-Dimethyl-2'-(3-methyl-butylca...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123510(2'-[(3-Phenyl-butyrylamino)-methyl]-biphenyl-2-car...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123529(CHEMBL147039 | [6,6'-Dimethyl-2'-(3-methyl-butylca...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123530(CHEMBL147315 | [2'-(2,4-Difluoro-benzylcarbamoyl)-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123519(2'-{[2-(4-Methoxy-phenyl)-acetylamino]-methyl}-bip...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123531(CHEMBL147962 | [2'-(3-Dimethylamino-2,2-dimethyl-p...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123508(CHEMBL148159 | [2'-(2-Pyridin-2-yl-ethylcarbamoyl)...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.3 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123524(CHEMBL146771 | [2'-(2-Pyridin-2-yl-ethylcarbamoyl)...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123533(2'-(Benzenesulfonylamino-methyl)-biphenyl-2-carbox...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123516(CHEMBL144170 | {2-[2-(3-Methyl-butylcarbamoyl)-pyr...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123515(CHEMBL144106 | [2'-(3-Methyl-butylcarbamoyl)-biphe...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123512(CHEMBL148258 | [2'-(3-Methyl-butylcarbamoyl)-biphe...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123513(2'-(Phenethylamino-methyl)-biphenyl-2-carboxylic a...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123534(2'-(Benzoylamino-methyl)-biphenyl-2-carboxylic aci...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123522(2'-[(3-Phenyl-ureido)-methyl]-biphenyl-2-carboxyli...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123527(2'-[(3-Trifluoromethyl-benzenesulfonylamino)-methy...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123517(CHEMBL358048 | {4-[2-(3-Methyl-butylcarbamoyl)-phe...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123523(CHEMBL146772 | [2'-(3-Methyl-butylcarbamoyl)-biphe...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123509(2'-[(4-Acetyl-benzenesulfonylamino)-methyl]-biphen...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123526(CHEMBL143727 | {2-[3-(3-Methyl-butylcarbamoyl)-pyr...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123514(2'-[(Naphthalene-1-sulfonylamino)-methyl]-biphenyl...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123520(8-(4-Chloro-benzenesulfonylamino)-naphthalene-1-ca...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123532(2'-[(Naphthalene-1-sulfonylamino)-methyl]-biphenyl...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 5(Homo sapiens (Human))
Aventis Pharma Deutschland

Curated by ChEMBL
LigandPNGBDBM50123535(CHEMBL146726 | {2-[4-(3-Methyl-butylcarbamoyl)-pyr...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed