Compile Data Set for Download or QSAR
maximum 50k data
Found 41 Enz. Inhib. hit(s) with all data for entry = 50035362
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124310(CHEMBL170406 | Sodium; 4-{4-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124307(2-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124308(CHEMBL173484 | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124335(2-Amino-N-{3-[2-amino-3-cyano-6-(2-hydroxy-phenyl)...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124323(3-Amino-N-{3-[2-amino-3-cyano-6-(2-hydroxy-phenyl)...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124327(4-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124336(CHEMBL424766 | Sodium; 2-[2-amino-3-cyano-6-(2-hyd...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124312(CHEMBL354947 | Sodium; 4-[2-amino-3-cyano-6-(2-hyd...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124309(CHEMBL535135 | N-{5-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  800nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124319(CHEMBL434691 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50:  900nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124316(CHEMBL171291 | N-{4-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124306(CHEMBL534692 | N-{5-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124337(CHEMBL174201 | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124324(CHEMBL170189 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124313(5-Oxo-tetrahydro-furan-2-carboxylic acid {3-[2-ami...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124317(CHEMBL366730 | Sodium; 4-{3-[2-amino-3-cyano-6-(5-...)
Affinity DataIC50:  1.70E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124330(3-[2-Amino-3-cyano-6-(2-hydroxy-phenyl)-pyridin-4-...)
Affinity DataIC50:  1.80E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124315(CHEMBL173111 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50:  2.00E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124326(CHEMBL558038 | N-{5-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124305(CHEMBL440200 | Sodium; 3-[2-amino-3-cyano-6-(2-hyd...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124331(CHEMBL262056 | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  3.00E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124314(CHEMBL173747 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50:  5.30E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124339(CHEMBL174430 | Sodium; 4-{3-[2-amino-6-(5-chloro-2...)
Affinity DataIC50:  5.50E+3nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124338(CHEMBL1187917 | CHEMBL534462 | N-{3-[2-Acetylamino...)
Affinity DataIC50:  1.50E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124334(CHEMBL444345 | Sodium; 4-[3-(2-amino-3-cyano-6-phe...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124320(2-Amino-4-(3-amino-phenyl)-6-(2-hydroxy-phenyl)-ni...)
Affinity DataIC50:  2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124313(5-Oxo-tetrahydro-furan-2-carboxylic acid {3-[2-ami...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human IKK-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124318(CHEMBL424000 | Sodium; 4-{3-[2-amino-3-cyano-6-(4-...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124308(CHEMBL173484 | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human mitogen-activated protein kinase kinase 4 (MKK4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124332(CHEMBL170355 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124308(CHEMBL173484 | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124333(CHEMBL171680 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124321(CHEMBL535358 | N-{3-[2-Amino-3-cyano-6-(3-hydroxy-...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124325(CHEMBL535359 | N-{3-[3-Cyano-2-hydroxy-6-(2-hydrox...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit alpha(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124308(CHEMBL173484 | N-{3-[2-Amino-3-cyano-6-(2-hydroxy-...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human IKK-alpha kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124313(5-Oxo-tetrahydro-furan-2-carboxylic acid {3-[2-ami...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human mitogen-activated protein kinase kinase 4 (MKK4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124322(CHEMBL539837 | N-{3-[3-Cyano-2-diethylamino-6-(2-h...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124311(2-Amino-4-(4-dimethylamino-phenyl)-6-(2-hydroxy-ph...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124313(5-Oxo-tetrahydro-furan-2-carboxylic acid {3-[2-ami...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human SykMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124329(2-Amino-6-(2-hydroxy-phenyl)-4-(4-nitro-phenyl)-ni...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Kyoto 619-0216

Curated by ChEMBL
LigandPNGBDBM50124328(CHEMBL171587 | Sodium; 4-{3-[2-amino-3-cyano-6-(2-...)
Affinity DataIC50: >2.00E+4nMAssay Description:In vitro inhibitory concentration required against recombinant human IkB kinase beta (IKK-beta)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed