Affinity Data by PubMed id=1317407

PubMed code 1317407

Found 7 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Nociceptin/mu opioid receptor (Rattus norvegicus (rat))	BDBM50000296 (CHEMBL441765 \| CHEMBL482811 \| U-50488H) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar	Purchase CHEBI CHEMBL KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Nociceptin/mu opioid receptor (Rattus norvegicus (rat))	BDBM50292538 ((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...) Show SMILES CN1CC[C@]2(C)[C@H]1N(C)c1ccc(O)cc21 Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar	Purchase CHEBI CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Nociceptin/mu opioid receptor (Rattus norvegicus (rat))	BDBM50292537 (CHEMBL484665 \| akuammine) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Nociceptin/mu opioid receptor (Rattus norvegicus (rat))	BDBM50292540 (CHEMBL489955 \| dihydroakuammine) Show SMILES Show InChI	PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	6.00E+3	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Opioid receptors; mu & delta (Rattus norvegicus (rat))	BDBM50292538 ((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...) Show SMILES CN1CC[C@]2(C)[C@H]1N(C)c1ccc(O)cc21 Show InChI	PDB Reactome pathway KEGG B.MOAD GoogleScholar	Purchase CHEBI CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	1.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]pCl-DPDP from delta opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Opioid receptors; mu & delta (Rattus norvegicus (rat))	BDBM50292537 (CHEMBL484665 \| akuammine) Show SMILES Show InChI	PDB Reactome pathway KEGG B.MOAD GoogleScholar	CHEMBL KEGG PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.00E+4	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]pCl-DPDP from delta opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair
Opioid receptors; mu & delta (Rattus norvegicus (rat))	BDBM50292540 (CHEMBL489955 \| dihydroakuammine) Show SMILES Show InChI	PDB Reactome pathway KEGG B.MOAD GoogleScholar	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	>1.00E+5	n/a	n/a	n/a	n/a	n/a	n/a
TBA Curated by ChEMBL					Assay Description Displacement of [3H]pCl-DPDP from delta opioid receptor in rat central nervous system membrane				J Nat Prod 55: 380-384 (1992) Article DOI: 10.1021/np50081a017 BindingDB Entry DOI: 10.7270/Q28W3DBN
TBA Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%