Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet activating factor receptor (Cavia porcellus) | BDBM50000714![]() (3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000717![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 142 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000701![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 157 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000707![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 167 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000722![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 331 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000720![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-di...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 345 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000719![]() (CHEMBL62812 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000708![]() (4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 656 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000700![]() (4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000716![]() (CHEMBL61680 | {7-[4-(4-Fluoro-phenyl)-1-methyl-but...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 925 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000718![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 945 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000705![]() (2-({7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydro...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000712![]() (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-dimet...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.25E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000711![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000715![]() (2-[7-(1,2-Dimethyl-heptyl)-5-hydroxy-10,10-dimethy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000702![]() (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methoxy-1...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.21E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000710![]() (3-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000699![]() (3-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000709![]() (5-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000724![]() (2-(5-Hydroxy-7-isopropyl-10,10-dimethyl-1,2,4,10-t...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000725![]() (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-10,10-dimet...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.18E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000721![]() (2-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000703![]() (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methoxy-1...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.69E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000723![]() (1-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.05E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000726![]() (4-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-hydrox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000713![]() (2-[5-{4-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-2,6-d...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.35E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000706![]() (6-{7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-5-methox...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet activating factor receptor (Cavia porcellus) | BDBM50000704![]() (7-[4-(4-Fluoro-phenyl)-1-methyl-butyl]-1,4,4-trime...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar | CHEMBL PC cid PC sid UniChem | Article PubMed | 4.38E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Abbott Laboratories Curated by ChEMBL | Assay Description In vitro intrinsic binding affinity at platelet activating factor receptor using rabbit platelet membranes | J Med Chem 35: 2055-61 (1992) Article DOI: 10.1021/jm00089a016 BindingDB Entry DOI: 10.7270/Q2NZ86K9 | |||||||||||
More data for this Ligand-Target Pair |