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Found 14 Enz. Inhib. hit(s) with all data for entry = 4657
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81541(CAS_195530 | NSC_195530 | S-Beta-Dimethylhistamine...)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81541(CAS_195530 | NSC_195530 | S-Beta-Dimethylhistamine...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81543(Alpha-Dimethylhistane-alpha | CAS_195960 | NSC_195...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM22904((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81542(Beta-Methylhistamine | CAS_565544 | NSC_565544)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81542(Beta-Methylhistamine | CAS_565544 | NSC_565544)
Affinity DataKi:  0.900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM22904((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...)
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81543(Alpha-Dimethylhistane-alpha | CAS_195960 | NSC_195...)
Affinity DataKi:  270nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81542(Beta-Methylhistamine | CAS_565544 | NSC_565544)
Affinity DataKi:  282nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM22904((2R)-1-(1H-imidazol-5-yl)propan-2-amine | (R)-alph...)
Affinity DataKi:  1.55E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Queen'S Medical Centre

Curated by PDSP Ki Database
LigandPNGBDBM81541(CAS_195530 | NSC_195530 | S-Beta-Dimethylhistamine...)
Affinity DataKi:  1.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed