Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 5739
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92971(Amphiphile, VI)
Affinity DataIC50:  1.10E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92969(Amphiphile, IV)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92976(Amphiphile, XI)
Affinity DataIC50:  1.50E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92978(Amphiphile, XIII)
Affinity DataIC50:  2.00E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92979(Amphiphile, XVI)
Affinity DataIC50:  2.60E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92980(Amphiphile, XVII)
Affinity DataIC50:  4.00E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92974(Amphiphile, IX)
Affinity DataIC50:  5.90E+4nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92977(Amphiphile, XII)
Affinity DataIC50:  1.64E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92973(Amphiphile, VIII)
Affinity DataIC50:  1.91E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92972(Amphiphile, VII)
Affinity DataIC50:  2.46E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92968(Amphiphile, III)
Affinity DataIC50:  2.58E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92975(Amphiphile, X)
Affinity DataIC50:  4.08E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Mcmaster University

LigandPNGBDBM92970(Amphiphile, V)
Affinity DataIC50:  6.43E+5nMpH: 7.5 T: 2°CAssay Description:The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed