Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50036048
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075539(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-[1,2,4]thia...)
Affinity DataIC50:  11nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003117(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-4H-[1,2,4]o...)
Affinity DataIC50:  50nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003122(4-(5-Aminomethyl-[1,2,4]thiadiazol-3-yl)-2,6-di-te...)
Affinity DataIC50:  87nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003124(2,6-Di-tert-butyl-4-(3-chloromethyl-[1,2,4]oxadiaz...)
Affinity DataIC50:  100nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012896(CHEMBL876 | CL-583.NA SALT | MECLOFENAMATE SODIUM ...)
Affinity DataIC50:  100nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003110(CHEMBL543891 | N-[3-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  140nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003121(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-dihydro-fur...)
Affinity DataIC50:  150nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003123(1-[3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-[1,2,4]t...)
Affinity DataIC50:  170nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003111(2,6-Di-tert-butyl-4-(5-methyl-[1,2,4]oxadiazol-3-y...)
Affinity DataIC50:  300nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003126(4-(5-Amino-[1,2,4]thiadiazol-3-yl)-2,6-di-tert-but...)
Affinity DataIC50:  330nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003125(CHEMBL542464 | N-[3-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  370nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003109(2,6-Di-tert-butyl-4-(3-dimethylaminomethyl-[1,2,4]...)
Affinity DataIC50:  450nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003114(2,6-Di-tert-butyl-4-(3-methyl-[1,2,4]oxadiazol-5-y...)
Affinity DataIC50:  460nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003116(CHEMBL331793 | N-[3-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  670nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003118(2,6-Di-tert-butyl-4-(5-dimethylaminomethyl-[1,2,4]...)
Affinity DataIC50:  730nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003124(2,6-Di-tert-butyl-4-(3-chloromethyl-[1,2,4]oxadiaz...)
Affinity DataIC50:  780nMAssay Description:Inhibitory activity against 5-LipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003127(CHEMBL122193 | CHEMBL1626562 | CHEMBL16659 | choli...)
Affinity DataIC50:  800nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003123(1-[3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-[1,2,4]t...)
Affinity DataIC50:  1.20E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003112(CHEMBL123210 | N-[5-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against 5-LipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003110(CHEMBL543891 | N-[3-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  1.60E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003116(CHEMBL331793 | N-[3-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  1.70E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003113(4-(3-Amino-[1,2,4]oxadiazol-5-yl)-2,6-di-tert-buty...)
Affinity DataIC50:  1.90E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075539(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-[1,2,4]thia...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against 5-LipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003126(4-(5-Amino-[1,2,4]thiadiazol-3-yl)-2,6-di-tert-but...)
Affinity DataIC50:  2.20E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003111(2,6-Di-tert-butyl-4-(5-methyl-[1,2,4]oxadiazol-3-y...)
Affinity DataIC50:  2.30E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003119(4-(5-Amino-[1,2,4]oxadiazol-3-yl)-2,6-di-tert-buty...)
Affinity DataIC50:  2.50E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003121(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-dihydro-fur...)
Affinity DataIC50:  2.50E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003122(4-(5-Aminomethyl-[1,2,4]thiadiazol-3-yl)-2,6-di-te...)
Affinity DataIC50:  2.60E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003127(CHEMBL122193 | CHEMBL1626562 | CHEMBL16659 | choli...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory activity against 5-LipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003119(4-(5-Amino-[1,2,4]oxadiazol-3-yl)-2,6-di-tert-buty...)
Affinity DataIC50:  3.00E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003114(2,6-Di-tert-butyl-4-(3-methyl-[1,2,4]oxadiazol-5-y...)
Affinity DataIC50:  3.30E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003117(3-(3,5-Di-tert-butyl-4-hydroxy-phenyl)-4H-[1,2,4]o...)
Affinity DataIC50:  3.40E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003113(4-(3-Amino-[1,2,4]oxadiazol-5-yl)-2,6-di-tert-buty...)
Affinity DataIC50:  3.60E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003125(CHEMBL542464 | N-[3-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  4.40E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230039(CHEMBL332103)
Affinity DataIC50:  4.70E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003109(2,6-Di-tert-butyl-4-(3-dimethylaminomethyl-[1,2,4]...)
Affinity DataIC50:  6.80E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1/2(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003112(CHEMBL123210 | N-[5-(3,5-Di-tert-butyl-4-hydroxy-p...)
Affinity DataIC50:  7.20E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against Prostaglandin G/H synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50003118(2,6-Di-tert-butyl-4-(5-dimethylaminomethyl-[1,2,4]...)
Affinity DataIC50:  7.70E+3nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50012896(CHEMBL876 | CL-583.NA SALT | MECLOFENAMATE SODIUM ...)
Affinity DataIC50:  2.40E+4nMAssay Description:Evaluated in vitro for its inhibitory activity against 5-lipoxygenaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed