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PubMed code 1433224

Compile data set for download or QSAR
Found 1 hit of Enzyme Inhibition Constant Data   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Sodium channel protein type I I alpha subunit


(Rattus norvegicus)		BDBM50003618
PNG
(1-{2-[Bis-(4-trifluoromethyl-phenyl)-methoxy]-ethy...)
Show SMILES OC(=O)C1=CCCN(CCOC(c2ccc(cc2)C(F)(F)F)c2ccc(cc2)C(F)(F)F)C1
Show InChI InChI=1S/C23H21F6NO3/c24-22(25,26)18-7-3-15(4-8-18)20(16-5-9-19(10-6-16)23(27,28)29)33-13-12-30-11-1-2-17(14-30)21(31)32/h2-10,20H,1,11-14H2,(H,31,32)
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PC cid
PC sid
UniChem

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Article
PubMed
n/an/a 1.00E+4n/an/an/an/an/an/a



Warner-Lambert Company

Curated by ChEMBL


Assay Description
Inhibition of veratridine-stimulated [14C]- guanidine influx into rat cortical slice

J Med Chem 35: 4238-48 (1992)


Article DOI: 10.1021/jm00100a032
BindingDB Entry DOI: 10.7270/Q2W66P09
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%