Affinity DataEC50: 1.40nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
Affinity DataEC50: 470nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 4 receptor (mMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 8.80nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 4 receptor (mMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 2.40E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 600nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 2.70E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 5 receptor (hMC5R)More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 520nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 4.40E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
Affinity DataEC50: 440nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataEC50: 1.60nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Neurocrine Biosciences
Curated by ChEMBL
Neurocrine Biosciences
Curated by ChEMBL
Affinity DataEC50: >3.00E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 1 receptor (hMC1R)More data for this Ligand-Target Pair
Affinity DataEC50: 7.60nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 4 receptor (mMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 170nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 680nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 110nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 2 receptor (mMC2R)More data for this Ligand-Target Pair
Affinity DataEC50: 6.10nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human melanocortin receptor-4 (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 650nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:In vitro cAMP accumulation in Y1 cells transfected with mouse Melanocortin 4 receptor (mMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 380nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 690nMAssay Description:Agonistic activity measured as inhibition of cAMP accumulation in HEK cells expressing human Melanocortin 4 receptor (hMC4R)More data for this Ligand-Target Pair
Affinity DataEC50: 1.40E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair