Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Adenosine A1 receptor (GUINEA PIG) | BDBM50368473![]() (CHEMBL607797) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5.75E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368492![]() (CHEMBL607798) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.63E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368486![]() (CHEMBL608668) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.37E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368480![]() (CHEMBL607590) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.91E+3 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368470![]() (CHEMBL607891) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.61E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368475![]() (CHEMBL608745) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.41E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368483![]() (CHEMBL607605) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.90E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50009530![]() (3-(4-{2-[6-Amino-9-(3,4-dihydroxy-5-hydroxymethyl-...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.12E+5 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368478![]() (CHEMBL610444) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368485![]() (CHEMBL611609) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.02E+3 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368487![]() (CHEMBL607508) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9.12E+3 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368476![]() (CHEMBL608448) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.17E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368471![]() (CHEMBL608174) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.17E+3 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368465![]() (CHEMBL608451) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.95E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368491![]() (CHEMBL610445) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 6.03E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368490![]() (CHEMBL607874) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.32E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368484![]() (CHEMBL607872) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.91E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368474![]() (CHEMBL608167) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.23E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368466![]() (CHEMBL611947) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.26E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368469![]() (CHEMBL609338) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.90E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368488![]() (CHEMBL611610) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.29E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368464![]() (CHEMBL608176) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.17E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368489![]() (CHEMBL611571) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.98E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368463![]() (CHEMBL608175) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 832 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368467![]() (CHEMBL607886) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368477![]() (CHEMBL607592) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 8.32E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368468![]() (CHEMBL607511) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.70E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368481![]() (CHEMBL607604) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.09E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368472![]() (CHEMBL611920) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 2.63E+3 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368479![]() (CHEMBL611918) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 4.17E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Adenosine A1 receptor (GUINEA PIG) | BDBM50368482![]() (CHEMBL608447) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 3.24E+4 | n/a | n/a | n/a | n/a |
University of South Florida Curated by ChEMBL | Assay Description Tested for adenosine A1 receptor agonistic activity by determining concentration needed to prolong the stimulus-QRS interval by 50% of the maximum re... | J Med Chem 35: 4562-6 (1993) Checked by Author Article DOI: 10.1021/jm00102a008 BindingDB Entry DOI: 10.7270/Q2CF9QQ1 | |||||||||||
More data for this Ligand-Target Pair |