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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Ionotropic glutamate receptor NMDA 1/2D (RAT) | BDBM83449 (1-(1-phenylcyclohexyl)piperidine;hydrochloride | M...) | PDB UniProtKB/SwissProt GoogleScholar | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ionotropic glutamate receptor NMDA 1/2D (RAT) | BDBM50004109 (1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 582 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ionotropic glutamate receptor NMDA 1/2D (RAT) | BDBM50004111 (1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 644 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ionotropic glutamate receptor NMDA 1/2D (RAT) | BDBM50004113 (1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 711 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM83449 (1-(1-phenylcyclohexyl)piperidine;hydrochloride | M...) | PDB UniProtKB/SwissProt GoogleScholar | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | 1.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50004112 (1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50004113 (1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.72E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50004109 (1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.45E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50004110 (1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.28E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ionotropic glutamate receptor NMDA 1/2D (RAT) | BDBM50004112 (1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8.22E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50004111 (1-(3-Phenyl-bicyclo[3.1.0]hex-3-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-(+)-pentazocine from sigma receptor in Guinea pig brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Ionotropic glutamate receptor NMDA 1/2D (RAT) | BDBM50004110 (1-(2-Phenyl-bicyclo[3.1.0]hex-2-yl)-piperidine | C...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Diabetes and Digestive and Kidney Diseases Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor in rat brain | J Med Chem 35: 4704-12 (1993) Article DOI: 10.1021/jm00103a008 BindingDB Entry DOI: 10.7270/Q2NP23CB | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
