Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50004169![]() ((2S,3S)-3-(4-Chloro-phenyl)-8-methyl-2-vinyl-8-aza...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Mayo Foundation Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]mazindol binding from rat striatal membranes | J Med Chem 35: 4764-6 (1993) Article DOI: 10.1021/jm00103a015 BindingDB Entry DOI: 10.7270/Q2QR4XQT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50035738![]() ((R)-3-(4-Chloro-phenyl)-8-methyl-8-aza-bicyclo[3.2...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Mayo Foundation Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]mazindol binding from rat striatal membranes | J Med Chem 35: 4764-6 (1993) Article DOI: 10.1021/jm00103a015 BindingDB Entry DOI: 10.7270/Q2QR4XQT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50004170![]() (Benzoic acid 2-(2-chloro-vinyl)-8-methyl-8-aza-bic...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 222 | n/a | n/a | n/a | n/a | n/a | n/a |
Mayo Foundation Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]mazindol binding from rat striatal membranes | J Med Chem 35: 4764-6 (1993) Article DOI: 10.1021/jm00103a015 BindingDB Entry DOI: 10.7270/Q2QR4XQT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM22418![]() (Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase CHEBI DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 580 | n/a | n/a | n/a | n/a | n/a | n/a |
Mayo Foundation Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]mazindol binding from rat striatal membranes | J Med Chem 35: 4764-6 (1993) Article DOI: 10.1021/jm00103a015 BindingDB Entry DOI: 10.7270/Q2QR4XQT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Sodium-dependent dopamine transporter (Rattus norvegicus (rat)) | BDBM50004168![]() (Benzoic acid 8-methyl-2-vinyl-8-aza-bicyclo[3.2.1]...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.73E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Mayo Foundation Curated by ChEMBL | Assay Description Compound was evaluated for its ability to displace [3H]mazindol binding from rat striatal membranes | J Med Chem 35: 4764-6 (1993) Article DOI: 10.1021/jm00103a015 BindingDB Entry DOI: 10.7270/Q2QR4XQT | |||||||||||
More data for this Ligand-Target Pair |