Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with all data for entry = 50014090
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50:  38nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50:  74nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human activated protein C (APC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human alpha-thrombin (FIIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human tissue type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >130nMAssay Description:Compound was tested for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human tissue type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human activated protein C (APC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50: >170nMAssay Description:Compound was tested for inhibition of human alpha-thrombin (FIIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138161(CHEMBL321466 | N-{1-[(3-Aminomethyl-phenylcarbamoy...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50:  250nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138156(Biphenyl-4-carboxylic acid {1-[(3-aminomethyl-phen...)
Affinity DataIC50: >250nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50:  330nMAssay Description:Compound was tested for inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50:  360nMAssay Description:Compound was tested for inhibition of human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human tissue type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human activated protein C (APC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138154(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-me...)
Affinity DataIC50: >450nMAssay Description:Compound was tested for inhibition of human alpha-thrombin (FIIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50: >870nMAssay Description:Compound was tested for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50: >870nMAssay Description:Compound was tested for inhibition of human urokinase-type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50: >870nMAssay Description:Compound was tested for inhibition of human alpha-thrombin (FIIa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50: >870nMAssay Description:Compound was tested for inhibition of human activated protein C (APC)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50138157(Biphenyl-4-carboxylic acid {1-[(5-aminomethyl-2-ch...)
Affinity DataIC50: >870nMAssay Description:Compound was tested for inhibition of human tissue type plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204029(CHEMBL419366)
Affinity DataIC50:  890nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204638(CHEMBL320473)
Affinity DataIC50:  980nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204631(CHEMBL432789)
Affinity DataIC50:  980nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204028(CHEMBL104220)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50206966(CHEMBL322441)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204634(CHEMBL320722)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50207118(CHEMBL320659)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204069(CHEMBL107427)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204033(CHEMBL317458)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50206960(CHEMBL106903)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204044(CHEMBL104601)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204036(CHEMBL326694)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204636(CHEMBL106146)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204943(CHEMBL104309)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204637(CHEMBL319925)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204038(CHEMBL107791)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204045(CHEMBL106183)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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