TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 76nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 183nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 255nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 323nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 503nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 540nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 659nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 682nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 3(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory potency against MAP kinase kinase 3 (MKK3)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceuticals Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibitory potency against mitogen activated protein kinase kinase kinase 1More data for this Ligand-Target Pair