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Found 22 Enz. Inhib. hit(s) with all data for entry = 50014440
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142763(CHEMBL50184 | [3-Chloro-5-({6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  1.40nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142773((3-Chloro-5-{[6-[2-(5-ethyl-4-methyl-thiazol-2-yl)...)
Affinity DataIC50:  4.40nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50404353(CHEMBL2113710)
Affinity DataIC50:  4.70nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142770((3-Chloro-5-{[6-[2-(5-ethyl-4-methyl-thiazol-2-yl)...)
Affinity DataIC50:  5.5nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142762((3-Chloro-5-{[6-[2-(5-ethyl-4-methyl-thiazol-2-yl)...)
Affinity DataIC50:  6.5nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142761((3-Chloro-5-{[6-[2-(5-ethyl-4-methyl-thiazol-2-yl)...)
Affinity DataIC50:  8.40nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142782(CHEMBL264820 | [3-Chloro-5-({4-cyclopentyloxy-6-[2...)
Affinity DataIC50:  11nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142769(CHEMBL52282 | [3-Chloro-5-({4-cyclobutoxy-6-[2-(5-...)
Affinity DataIC50:  11nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142775(CHEMBL298983 | [3-Chloro-5-({6-[2-(5-ethyl-4-methy...)
Affinity DataIC50:  12nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142779(CHEMBL48950 | [3-({4-Butoxy-6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  16nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142771((3-Chloro-5-{[6-[2-(5-ethyl-4-methyl-thiazol-2-yl)...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142766(CHEMBL299598 | [3-Chloro-5-({6-[2-(5-ethyl-4-methy...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142764((3-Chloro-5-{[6-[2-(5-ethyl-4-methyl-thiazol-2-yl)...)
Affinity DataIC50:  20nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142777(CHEMBL49461 | [3-Chloro-5-({4-cyclohexyloxy-6-[2-(...)
Affinity DataIC50:  29nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142772(CHEMBL48897 | [3-Chloro-5-({6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  30nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142781(CHEMBL48947 | [3-Chloro-5-({4-ethoxy-6-[2-(5-ethyl...)
Affinity DataIC50:  33nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142774(CHEMBL48456 | [3-Chloro-5-({6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  35nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142768(CHEMBL422583 | [3-Chloro-5-({4-(2,2-dimethyl-propo...)
Affinity DataIC50:  55nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142765(CHEMBL51422 | [3-Chloro-5-({6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  63nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142780(CHEMBL48493 | [3-Chloro-5-({6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  72nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142778(CHEMBL49795 | [3-Chloro-5-({6-[2-(5-ethyl-4-methyl...)
Affinity DataIC50:  234nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50142767(CHEMBL45869 | [3-({4-Benzyloxy-6-[2-(5-ethyl-4-met...)
Affinity DataIC50:  237nMAssay Description:Binding affinity against human recombinant NPY Y1 receptor in CHO/dhFr- cell membranes using [125I]-PYYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed