Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 1891
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM14824(4-({5-bromo-4-[(4-methoxyphenyl)amino]pyrimidin-2-...)
Affinity DataIC50:  450nMpH: 7.5 T: 2°CAssay Description:The compound inhibitory activity was determined by incubation with purified recombinant Chk1 and biotinylated peptide substrate in the presence ATP/[...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM14825(3-[7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]-2-o...)
Affinity DataIC50:  4.00E+3nMpH: 7.5 T: 2°CAssay Description:The compound inhibitory activity was determined by incubation with purified recombinant Chk1 and biotinylated peptide substrate in the presence ATP/[...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed