Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50035399
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Upr 2301 Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50147700((1H-Indol-2-ylmethyl)-(1-naphthalen-1-yl-ethyl)-am...)
Affinity DataEC50:  1.30E+3nMAssay Description:Ability to stimulate [3H]inositol phosphates accumulation in CHO cells expressing rat Calcium sensing receptor (CaSR) at 2 mM [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Rattus norvegicus)
Upr 2301 Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50404271(CHEMBL2092942)
Affinity DataEC50:  1.00E+3nMAssay Description:Ability to stimulate [3H]inositol phosphates accumulation in CHO cells expressing rat Calcium sensing receptor (CaSR) at 2 mM [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Upr 2301 Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50404271(CHEMBL2092942)
Affinity DataEC50:  310nMAssay Description:Ability to stimulate [3H]inositol phosphates accumulation in HEK293 cells expressing the human calcium sensing receptor (CaSR) at 2 mM [Ca2+]More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed