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Found 20 Enz. Inhib. hit(s) with all data for entry = 50042233
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157050(CHEMBL361914 | [4-(1-{2-[3-Methoxy-4-(3-o-tolyl-ur...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157041(CHEMBL185571 | [4-(1-{2-[3-Methoxy-4-(3-o-tolyl-ur...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157039(CHEMBL179780 | [4-(1-{2-[3-Methoxy-4-(3-o-tolyl-ur...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157044(CHEMBL369731 | [1-(1-{2-[4-(3-o-Tolyl-ureido)-phen...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157046(4-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pyr...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157048(CHEMBL360163 | [1-(4-{2-[4-(3-o-Tolyl-ureido)-phen...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157034(5-(3-Methyl-butylcarbamoyl)-5-[(1-{2-[4-(3-o-tolyl...)
Affinity DataIC50:  4.70nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157035(5-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pyr...)
Affinity DataIC50:  7.10nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157040(5-[(3-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-thi...)
Affinity DataIC50:  10nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157051(CHEMBL181708 | [4-(1-{2-[4-(3-o-Tolyl-ureido)-phen...)
Affinity DataIC50:  13nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157053(CHEMBL180106 | [4-(1-{2-[4-(3-o-Tolyl-ureido)-phen...)
Affinity DataIC50:  14nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157043(5-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-2,5...)
Affinity DataIC50:  20nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157047(5-[(4-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-mor...)
Affinity DataIC50:  26nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157037(5-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pip...)
Affinity DataIC50:  32nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157038(4-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pyr...)
Affinity DataIC50:  76nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157036(3-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pyr...)
Affinity DataIC50:  82nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157049(4-{[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-py...)
Affinity DataIC50:  121nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157052(1-(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pyrr...)
Affinity DataIC50:  148nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157045(6-[(1-{2-[4-(3-o-Tolyl-ureido)-phenyl]-acetyl}-pyr...)
Affinity DataIC50:  295nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-4/beta-1(Homo sapiens (Human))
Daiichi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50157042(CHEMBL182400 | [(1-{2-[4-(3-o-Tolyl-ureido)-phenyl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of VLA-4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed