Compile Data Set for Download or QSAR
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Found 32 Enz. Inhib. hit(s) with all data for entry = 50041391
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410165(CHEMBL372661)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410153(CHEMBL197216)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410158(CHEMBL195195)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410153(CHEMBL197216)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410165(CHEMBL372661)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410154(CHEMBL370969)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410156(CHEMBL195143)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410158(CHEMBL195195)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410152(CHEMBL371047)
Affinity DataIC50:  2.50E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410164(CHEMBL194829)
Affinity DataIC50:  2.62E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410156(CHEMBL195143)
Affinity DataIC50:  2.72E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50164888(6-Hydroxy-3-[1-(4-hydroxy-phenyl)-meth-(E)-ylidene...)
Affinity DataIC50:  3.07E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410152(CHEMBL371047)
Affinity DataIC50:  3.27E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410155(CHEMBL372372)
Affinity DataIC50:  3.51E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410163(CHEMBL364033)
Affinity DataIC50:  3.92E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410157(CHEMBL191658)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410160(CHEMBL381195)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50164888(6-Hydroxy-3-[1-(4-hydroxy-phenyl)-meth-(E)-ylidene...)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410154(CHEMBL370969)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410159(CHEMBL426092)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410151(CHEMBL381410)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410161(CHEMBL191804)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410162(CHEMBL193628)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410164(CHEMBL194829)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410163(CHEMBL364033)
Affinity DataIC50: >4.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase II activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410159(CHEMBL426092)
Affinity DataIC50:  5.55E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410155(CHEMBL372372)
Affinity DataIC50:  6.30E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410160(CHEMBL381195)
Affinity DataIC50:  8.00E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410151(CHEMBL381410)
Affinity DataIC50:  9.60E+5nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410157(CHEMBL191658)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410161(CHEMBL191804)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Kumamoto University

Curated by ChEMBL
LigandPNGBDBM50410162(CHEMBL193628)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibitory concentration against DNA topoisomerase I activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed