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Found 26 Enz. Inhib. hit(s) with all data for entry = 50016306
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50162116(2-(4-(benzyloxy)phenyl)-N-(1-(2-(pyrrolidin-1-yl)e...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory concentration against Melanin-concentrating hormone receptor 1 in diet-induced obese miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167565(1-[1-(2-Isobutylamino-ethyl)-1H-indazol-5-yl]-3-(4...)
Affinity DataIC50:  1.80nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167552(1-[1-(2-Cyclopentylamino-ethyl)-1H-indazol-5-yl]-3...)
Affinity DataIC50:  2.40nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167554(1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  5.90nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167561(1-[1-(3-Cyclopentylamino-propyl)-1H-indazol-5-yl]-...)
Affinity DataIC50:  8.5nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167567(1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167556(1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  19.8nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167558(1-[2-(4-Phenoxy-phenyl)-ethyl]-3-[1-(2-pyrrolidin-...)
Affinity DataIC50:  34.3nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167564(1-{1-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethy...)
Affinity DataIC50:  38.7nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167568(1-(3-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl...)
Affinity DataIC50:  40.6nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167550(1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-eth...)
Affinity DataIC50:  41.3nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167557(1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  78.5nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167553(1-{1-[3-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-prop...)
Affinity DataIC50:  82.9nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167569(1-{1-[3-(4-Hydroxy-piperidin-1-yl)-propyl]-1H-inda...)
Affinity DataIC50:  91.5nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167549(1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-eth...)
Affinity DataIC50:  113nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167571(1-(2-{5-[3-(4-Phenoxy-phenyl)-ureido]-indazol-1-yl...)
Affinity DataIC50:  134nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167563(2-(4-Phenoxy-benzylamino)-N-[1-(2-pyrrolidin-1-yl-...)
Affinity DataIC50:  299nMAssay Description:Inhibitory concentration against Melanin-concentrating hormone receptor 1 in diet-induced obese miceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167551(1-{1-[2-(3,3-Difluoro-pyrrolidin-1-yl)-ethyl]-1H-i...)
Affinity DataIC50:  305nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167548(1-(4-Phenoxy-benzyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  508nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167560(1-[2-(4-Phenoxy-phenyl)-ethyl]-3-[1-(2-pyrrolidin-...)
Affinity DataIC50:  545nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167566(1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  581nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167570(1-(1-Benzyl-piperidin-4-yl)-3-[1-(2-pyrrolidin-1-y...)
Affinity DataIC50:  971nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167572(1-(4-Benzyloxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-eth...)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167562(1-(4-Phenoxy-phenyl)-3-[1-(2-pyrrolidin-1-yl-ethyl...)
Affinity DataIC50:  1.85E+3nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167555(1-(1-Benzyl-piperidin-4-yl)-3-[1-(2-pyrrolidin-1-y...)
Affinity DataIC50:  4.51E+3nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50167559(1-{1-[2-(4-Hydroxy-piperidin-1-yl)-ethyl]-1H-indaz...)
Affinity DataIC50:  6.13E+3nMAssay Description:Inhibitory concentration against mouse Melanin-concentrating hormone receptor 1 expressed in IMR-32 cells using [125I]-MCHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed