Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 50016329
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167783(CHEMBL196885 | Decanoic acid {1-[3-(4-cyano-phenyl...)
Affinity DataIC50:  930nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167781(CHEMBL193448 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167778(CHEMBL194494 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167782(CHEMBL383346 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167784(CHEMBL197368 | Decanoic acid {1-[3-(3-cyano-phenyl...)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167780(CHEMBL370482 | Decanoic acid {1-[3-(2-cyano-phenyl...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167785(CHEMBL196248 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167786(CHEMBL371154 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 3(Homo sapiens (Human))
Vrije Universiteit Amsterdam

Curated by ChEMBL
LigandPNGBDBM50167779(CHEMBL371577 | Decanoic acid (2-dimethylamino-ethy...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory concentration against CX3C chemokine receptor 3 expressed in human HEK-293 cells using [125I]-CXCL10 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed