Compile Data Set for Download or QSAR
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Found 24 Enz. Inhib. hit(s) with all data for entry = 50037523
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170966(10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  2.44nMAssay Description:Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50026682(10-hydroxy-3,4-dimethoxy-17-methyl-(10S)-17-azatet...)
Affinity DataKi:  3.88nMAssay Description:Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50026687(3-hydroxy-4,10-dimethoxy-17-methyl-(10S)-17-azatet...)
Affinity DataKi:  4.65nMAssay Description:Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170964(3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  5.38nMAssay Description:Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  6.55nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170962(3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  31.7nMAssay Description:Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170963(3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  32.6nMAssay Description:Displacement of [3H][DAMGO] from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50370595(OXYCODONE | Oxycontin | US1184575, oxycodone | US9...)
Affinity DataKi:  43.6nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50026682(10-hydroxy-3,4-dimethoxy-17-methyl-(10S)-17-azatet...)
Affinity DataKi:  91.6nMAssay Description:Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170966(10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50026687(3-hydroxy-4,10-dimethoxy-17-methyl-(10S)-17-azatet...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170964(3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  197nMAssay Description:Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  217nMAssay Description:Displacement of [3H[Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170966(10-hydroxy-3,4-dimethoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  364nMAssay Description:Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170964(3-hydroxy-4,10-dimethoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  378nMAssay Description:Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170962(3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  498nMAssay Description:Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50026687(3-hydroxy-4,10-dimethoxy-17-methyl-(10S)-17-azatet...)
Affinity DataKi:  592nMAssay Description:Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50026682(10-hydroxy-3,4-dimethoxy-17-methyl-(10S)-17-azatet...)
Affinity DataKi:  693nMAssay Description:Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170963(3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  763nMAssay Description:Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170963(3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  881nMAssay Description:Displacement of [3H]Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50370595(OXYCODONE | Oxycontin | US1184575, oxycodone | US9...)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [3H[Ile5,6]-deltorphin II from delta opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50170962(3,10-dihydroxy-4-methoxy-17-methyl-17-azatetracycl...)
Affinity DataKi:  1.65E+3nMAssay Description:Displacement of[3H]U69,593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50370595(OXYCODONE | Oxycontin | US1184575, oxycodone | US9...)
Affinity DataKi:  2.66E+3nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed