Compile Data Set for Download or QSAR
maximum 50k data
Found 56 Enz. Inhib. hit(s) with all data for entry = 50017443
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182237(CHEMBL207947 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182245(CHEMBL437509 | N-((R)-6-((isobutylamino)methyl)-1,...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182221(CHEMBL381366 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182230(2-((S)-1-(benzo[b]thiophen-3-ylsulfonyl)piperidin-...)
Affinity DataIC50:  14nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182231(CHEMBL381979 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182222(CHEMBL380117 | N-((R)-6-((cyclopropylmethylamino)m...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182237(CHEMBL207947 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182220(CHEMBL381372 | N-((R)-6-((2-methoxyethylamino)meth...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182231(CHEMBL381979 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182221(CHEMBL381366 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  23nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182222(CHEMBL380117 | N-((R)-6-((cyclopropylmethylamino)m...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182245(CHEMBL437509 | N-((R)-6-((isobutylamino)methyl)-1,...)
Affinity DataIC50:  42nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182220(CHEMBL381372 | N-((R)-6-((2-methoxyethylamino)meth...)
Affinity DataIC50:  46nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182232(CHEMBL205981 | N-((R)-6-((cyclopropylamino)methyl)...)
Affinity DataIC50:  47nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182232(CHEMBL205981 | N-((R)-6-((cyclopropylamino)methyl)...)
Affinity DataIC50:  48nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182234(CHEMBL439505 | N-((R)-6-((cyclobutylamino)methyl)-...)
Affinity DataIC50:  54nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182234(CHEMBL439505 | N-((R)-6-((cyclobutylamino)methyl)-...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182229(CHEMBL203174 | N-((R)-6-((neopentylamino)methyl)-1...)
Affinity DataIC50:  59nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182236(CHEMBL205501 | N-((R)-6-((dimethylamino)methyl)-1,...)
Affinity DataIC50:  62nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182230(2-((S)-1-(benzo[b]thiophen-3-ylsulfonyl)piperidin-...)
Affinity DataIC50:  66nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182228(CHEMBL206247 | N-((R)-6-((isopropylamino)methyl)-1...)
Affinity DataIC50:  72nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182241(CHEMBL381964 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  73nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182239(CHEMBL208387 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  93nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182225(CHEMBL206901 | N-((R)-7-((tert-butylamino)methyl)c...)
Affinity DataIC50:  95nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182228(CHEMBL206247 | N-((R)-6-((isopropylamino)methyl)-1...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182241(CHEMBL381964 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182239(CHEMBL208387 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  130nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182235(2-((S)-1-(benzo[c][1,2,5]thiadiazol-4-ylsulfonyl)p...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182225(CHEMBL206901 | N-((R)-7-((tert-butylamino)methyl)c...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182236(CHEMBL205501 | N-((R)-6-((dimethylamino)methyl)-1,...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182235(2-((S)-1-(benzo[c][1,2,5]thiadiazol-4-ylsulfonyl)p...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182238(CHEMBL207945 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  210nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182246(CHEMBL205227 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  220nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182229(CHEMBL203174 | N-((R)-6-((neopentylamino)methyl)-1...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182238(CHEMBL207945 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  360nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182246(CHEMBL205227 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  440nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182242(2-[(S)-1-(biphenyl-4-sulfonyl)-piperidin-2-yl]-N-[...)
Affinity DataIC50:  540nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182226(CHEMBL206541 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  560nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182224(2-((S)-1-(4-butoxyphenylsulfonyl)piperidin-2-yl)-N...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182247(CHEMBL205242 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  610nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182242(2-[(S)-1-(biphenyl-4-sulfonyl)-piperidin-2-yl]-N-[...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182227(CHEMBL207033 | N-((R)-6-((2,2,2-trifluoroethylamin...)
Affinity DataIC50:  700nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182223(CHEMBL204847 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  780nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182226(CHEMBL206541 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  810nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182240(CHEMBL206801 | N-((R)-7-((tert-butylamino)methyl)c...)
Affinity DataIC50:  960nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182233(CHEMBL377011 | N-((R)-6-(azetidin-1-ylmethyl)-1,2,...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182224(2-((S)-1-(4-butoxyphenylsulfonyl)piperidin-2-yl)-N...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182223(CHEMBL204847 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human B1 receptor by calcium influx functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182240(CHEMBL206801 | N-((R)-7-((tert-butylamino)methyl)c...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50182243(CHEMBL208386 | N-((R)-6-((tert-butylamino)methyl)-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human B1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: