Found 18 Enz. Inhib. hit(s) with all data for entry = 50034614 TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human GST-tagged CDK4-cyclin D1 using his-tagged Rb as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human GST-tagged CDK4-cyclin D1 using his-tagged Rb as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 1.97E+6nMAssay Description:Inhibition of human CDK1-GST-tagged cyclin B using his-tagged Rb as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 2.36E+6nMAssay Description:Inhibition of human CDK2-GST-tagged cyclin E using his-tagged Rb as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 3.04E+6nMAssay Description:Inhibition of human CDK1-GST-tagged cyclin B using his-tagged Rb as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 3.21E+6nMAssay Description:Inhibition of Src using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 3.48E+6nMAssay Description:Inhibition of Src using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 4.14E+6nMAssay Description:Inhibition of human CDK2-GST-tagged cyclin E using his-tagged Rb as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: >2.00E+7nMAssay Description:Inhibition of c-Met using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: >2.00E+7nMAssay Description:Inhibition of c-Met using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 2.00E+7nMAssay Description:Inhibition of IGF1R using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: 2.20E+7nMAssay Description:Inhibition of IGF1R using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+7nMAssay Description:Inhibition of insulin receptor using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.10E+7nMAssay Description:Inhibition of insulin receptor using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of Lck using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of Lck using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of ERK1 using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 3(Homo sapiens (Human))
University Of Queensland
Curated by ChEMBL
University Of Queensland
Curated by ChEMBL
Affinity DataIC50: >1.00E+8nMAssay Description:Inhibition of ERK1 using fluorescent substrate by IMAP assayMore data for this Ligand-Target Pair
