Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50041442
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184908(CHEMBL402661 | cypate-[(RGD)4-NH2]1)
Affinity DataIC50:  25.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184904(CHEMBL206344 | cyclo(RGDfV) (control))
Affinity DataIC50:  28.7nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184902(CHEMBL407126 | cyclo[RGDfK(cypate)])
Affinity DataIC50:  63.9nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184906(CHEMBL429568 | cypate-[(RGD)4-NH2]2)
Affinity DataIC50:  79.6nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184903(CHEMBL415188 | cypate-[(RGD)2-NH2]2)
Affinity DataIC50:  104nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184905(CHEMBL413898 | cypate-[(RGD)3-NH2]2)
Affinity DataIC50:  132nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184907(CHEMBL412767 | cypate-[(RGD)3-NH2]1)
Affinity DataIC50:  481nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50184909(CHEMBL438186 | cypate-[(RGD)2-NH2]1)
Affinity DataIC50:  730nMAssay Description:Displacement of [125I]echistatin from AlphaV-beta-3 integrin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed