Compile Data Set for Download or QSAR
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Found 18 Enz. Inhib. hit(s) with all data for entry = 50017928
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188534((H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) | ...)
Affinity DataKi:  0.158nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188537(CHEMBL208916 | H-Dmt-Tic-Glu-Dap(6DMN)-NH(2))
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188534((H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) | ...)
Affinity DataKi:  41.3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(CHEMBL219407 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S...)
Affinity DataKi:  252nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(CHEMBL219407 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S...)
Affinity DataKi:  668nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(CHEMBL207661 | H-Tyr-Pro-Dap(6DMN)-Phe-NH2)
Affinity DataKi:  839nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(CHEMBL207661 | H-Tyr-Pro-Dap(6DMN)-Phe-NH2)
Affinity DataKi:  3.42E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataKi:  5.94E+3nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188537(CHEMBL208916 | H-Dmt-Tic-Glu-Dap(6DMN)-NH(2))
Affinity DataKi:  7.88E+3nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188537(CHEMBL208916 | H-Dmt-Tic-Glu-Dap(6DMN)-NH(2))
Affinity DataIC50:  100nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(CHEMBL219407 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S...)
Affinity DataIC50:  120nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188535(CHEMBL219407 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-NH-(C=S...)
Affinity DataIC50:  200nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188534((H-Dmt-Tic-Glu-NH-(CH(2))(5)-CO-Dap(6DMN)-NH(2) | ...)
Affinity DataIC50:  244nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataIC50:  253nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataIC50:  300nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(CHEMBL207661 | H-Tyr-Pro-Dap(6DMN)-Phe-NH2)
Affinity DataIC50:  389nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188536(CHEMBL207661 | H-Tyr-Pro-Dap(6DMN)-Phe-NH2)
Affinity DataIC50:  500nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed