Affinity DataKi: 0.0210nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 0.0510nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 7.58nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 18.8nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 27.4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 31.9nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 924nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataKi: 2.77E+3nMAssay Description:Displacement of [3H]deltorphin II from delta opioid receptor in rat synaptosomes P2 fractionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.79nMAssay Description:Activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.93nMAssay Description:Activity at mu opioid receptor by guinea pig ileum assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25.8nMAssay Description:Activity at delta opioid receptor assessed as inhibition of muscle contraction in mouse vas deferens assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Activity at delta opioid receptor assessed as inhibition of muscle contraction in mouse vas deferens assayMore data for this Ligand-Target Pair