Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50019483
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205216((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205202(3-((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205133((2S)-1-{[(2S,4S)-4-propyl-2-pyrrolidinyl]carbonyl}...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205128((2S)-1-{[(2S,4S)-4-allyl-2-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205219((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205214((2S)-1-{[(2S,4R)-4-(2-hydroxyethyl)-2-pyrrolidinyl...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205200((2S)-1-{[(2S,4S)-4-(1-azetidinylcarbonyl)-2-pyrrol...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205209((2S)-1-{[(2S,4S)-4-(4-morpholinylcarbonyl)-2-pyrro...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205215((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  4.40nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205224(2-((3R,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205223((2S)-1-{[(2S,4S)-4-(4-thiomorpholinylcarbonyl)-2-p...)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205212((2S)-1-{[(2S,4S)-4-(1-piperidinylcarbonyl)-2-pyrro...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205210((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205208((2S)-1-{[(2S,4S)-4-(1-pyrrolidinylcarbonyl)-2-pyrr...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205213(2S)-1-{[(2S,4S,5S)-4-(1,3-dihydro-2H-isoindol-2-yl...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205221((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205218((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205222((2S)-1-{[(2S,4S,5S)-5-methyl-4-(4-thiomorpholinylc...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205217((2S)-1-{[(2S,4S)-4-(hydroxymethyl)-2-pyrrolidinyl]...)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205211((2S)-1-{[(2S,4S,5S)-5-Methyl-4-(1-pyrrolidinylcarb...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205204((3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}-...)
Affinity DataIC50:  7.70nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205203((2S)-1-{[(2S,4S)-4-(1-azepanylcarbonyl)-2-pyrrolid...)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205206((2S,3S,5S)-5-((S)-2-cyanopyrrolidine-1-carbonyl)-N...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205220((2S)-1-{[(2S,4S)-4-(1-azocanylcarbonyl)-2-pyrrolid...)
Affinity DataIC50:  11nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205226((2S)-1-{[(2S,4S,5S)-5-methyl-4-(1-piperidinylcarbo...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205207((2S)-1-{[(2S,4S,5S)-4-(1-azetidinylcarbonyl)-5-met...)
Affinity DataIC50:  13nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205205((2S,3S,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbony...)
Affinity DataIC50:  15nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205225(((3R,5S)-5-{[(2S)-2-cyano-1-pyrrolidinyl]carbonyl}...)
Affinity DataIC50:  16nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM11056((2S)-1-[(2S)-pyrrolidin-2-ylcarbonyl]pyrrolidine-2...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50205201((2S)-1-{[(2S,4S,5S)-5-methyl-4-(4-morpholinylcarbo...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed