Compile Data Set for Download or QSAR
maximum 50k data
Found 42 Enz. Inhib. hit(s) with all data for entry = 50020285
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212166(7-chloro-6H-chromeno[4,3-b]quinoline-3,9-diol | CH...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212173(7-bromo-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171724(4-Bromo-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-bro...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171726(4-Chloro-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-ch...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212172(3,9-dihydroxy-6H-chromeno[4,3-b]quinoline-7-carbon...)
Affinity DataIC50:  6.10nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212161(7-vinyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)
Affinity DataIC50:  22nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171712(6-Hydroxy-2-(4-hydroxy-phenyl)-quinoline-4-carboni...)
Affinity DataIC50:  28nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212162(7-ethyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)
Affinity DataIC50:  46nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171723(4-Ethyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-eth...)
Affinity DataIC50:  52nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212170(7-ethynyl-6H-chromeno[4,3-b]quinoline-3,9-diol | C...)
Affinity DataIC50:  52nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212173(7-bromo-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)
Affinity DataIC50:  56nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171727(2-(4-Hydroxy-phenyl)-4-vinyl-quinolin-6-ol | 2-(4-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212168(4-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)
Affinity DataIC50:  65nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171729(4-Ethynyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-e...)
Affinity DataIC50:  75nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212167(7-(3-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)
Affinity DataIC50:  86nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212166(7-chloro-6H-chromeno[4,3-b]quinoline-3,9-diol | CH...)
Affinity DataIC50:  88nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212163(7-(4-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)
Affinity DataIC50:  94nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212172(3,9-dihydroxy-6H-chromeno[4,3-b]quinoline-7-carbon...)
Affinity DataIC50:  98nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212165(7-(3-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)
Affinity DataIC50:  144nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212169(3-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212164(7-(4-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171724(4-Bromo-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-bro...)
Affinity DataIC50:  212nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171726(4-Chloro-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-ch...)
Affinity DataIC50:  213nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212171(7-(4-(trifluoromethyl)phenyl)-6H-chromeno[4,3-b]qu...)
Affinity DataIC50:  319nMAssay Description:Inhibition of human ERalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  395nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171712(6-Hydroxy-2-(4-hydroxy-phenyl)-quinoline-4-carboni...)
Affinity DataIC50:  455nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212165(7-(3-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)
Affinity DataIC50:  504nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171727(2-(4-Hydroxy-phenyl)-4-vinyl-quinolin-6-ol | 2-(4-...)
Affinity DataIC50:  504nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212161(7-vinyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)
Affinity DataIC50:  526nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212163(7-(4-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)
Affinity DataIC50:  549nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212170(7-ethynyl-6H-chromeno[4,3-b]quinoline-3,9-diol | C...)
Affinity DataIC50:  624nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171723(4-Ethyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-eth...)
Affinity DataIC50:  634nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212162(7-ethyl-6H-chromeno[4,3-b]quinoline-3,9-diol | CHE...)
Affinity DataIC50:  641nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212167(7-(3-methoxyphenyl)-6H-chromeno[4,3-b]quinoline-3,...)
Affinity DataIC50:  820nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212168(4-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212169(3-(3,9-dihydroxy-6H-chromeno[4,3-b]quinolin-7-yl)b...)
Affinity DataIC50:  1.13E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50171729(4-Ethynyl-2-(4-hydroxy-phenyl)-quinolin-6-ol | 4-e...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212164(7-(4-chlorophenyl)-6H-chromeno[4,3-b]quinoline-3,9...)
Affinity DataIC50:  2.35E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIsoform 1 of Steroid hormone receptor ERR2 (ERRbeta2-delta10)(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50212171(7-(4-(trifluoromethyl)phenyl)-6H-chromeno[4,3-b]qu...)
Affinity DataIC50:  5.24E+3nMAssay Description:Inhibition of human ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed