Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50025455
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50242614((S)-1-((S)-2-((S)-2,5-diamino-5-oxopentanamido)-3-...)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake after 1 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50242617(CHEMBL521026 | QSPac)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake after 1 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50242615(CHEMBL486028 | QCPac)
Affinity DataIC50:  2nMAssay Description:Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake after 1 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 1(Homo sapiens (Human))
University WüRzburg

Curated by ChEMBL
LigandPNGBDBM50242616(CHEMBL485831 | QCP)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human SGLT1 expressed in xenopus laevis oocyte assessed as inhibition of methyl-alpha-D-[14C]glucopyranoside uptake after 1 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed