Compile Data Set for Download or QSAR
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Found 31 Enz. Inhib. hit(s) with all data for entry = 50038266
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373021(CHEMBL401616)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373910(CHEMBL410704)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at mouse PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373906(CHEMBL272175)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373907(CHEMBL271394)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373908(CHEMBL407950)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373909(CHEMBL272466)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373910(CHEMBL410704)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373911(CHEMBL410705)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373912(CHEMBL270961)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373913(CHEMBL271776)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373914(CHEMBL271775)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373021(CHEMBL401616)
Affinity DataEC50:  1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373911(CHEMBL410705)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50:  1.00E+5nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  9.60E+3nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28700(2-(4-(4-Chlorobenzoyl)phenoxy)-2-methylpropionic a...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM28701(2-(4-{2-[(4-chlorophenyl)formamido]ethyl}phenoxy)-...)
Affinity DataEC50:  3.00E+4nMAssay Description:Agonist activity at human PPARdelta expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373915(CHEMBL272017)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373916(CHEMBL273036)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373917(CHEMBL273035)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373916(CHEMBL273036)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373917(CHEMBL273035)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373021(CHEMBL401616)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at mouse PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373907(CHEMBL271394)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50373910(CHEMBL410704)
Affinity DataEC50:  100nMAssay Description:Agonist activity at mouse PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Nippon Shinyaku

Curated by ChEMBL
LigandPNGBDBM50225835((2s,5s)-2-methyl-5-(4-(5-methyl-2-p-tolyloxazol-4-...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARalpha expressed in CV1 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed