Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50032224
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition of Saccharomyces cerevisiae Pho80-Pho85-Pho81-MD catalyzed phosphorylation of Pho4 assessed as increase in substrate concentra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphate system positive regulatory protein PHO81(Saccharomyces cerevisiae)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae Pho81-MD-dependent Pho80-Pho85 activity after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphate system positive regulatory protein PHO81(Saccharomyces cerevisiae)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae Pho81-MD-MD dependent Pho80-Pho85 activity after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphate system positive regulatory protein PHO81(Saccharomyces cerevisiae)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae Pho81-MD-dependent Pho80-Pho85 activity after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae Pho80-Pho85-Pho81-MD catalyzed phosphorylation of Pho4-site 6 peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphate system positive regulatory protein PHO81(Saccharomyces cerevisiae)
Harvard University

Curated by ChEMBL
LigandPNGBDBM50326018((1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentakis(phosphonoox...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of Saccharomyces cerevisiae Pho81-MD-MD dependent Pho80-Pho85 activity after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed