Compile Data Set for Download or QSAR
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Found 17 Enz. Inhib. hit(s) with all data for entry = 50022021
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230586(CHEMBL252845 | N-((2-amino-6-methylpyridin-3-yl)me...)
Affinity DataEC50:  15nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230602(CHEMBL252085 | N-(2-amino-6-methyl-pyridin-3-ylmet...)
Affinity DataEC50:  1.02E+5nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230588(3-(2-amino-6-methyl-pyridin-3-ylmethyl)-5-(2-hydro...)
Affinity DataEC50:  28nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230589(3-(2-amino-pyridin-3-ylmethyl)-5-(2-hydroxy-ethyl)...)
Affinity DataEC50:  110nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230590(CHEMBL402594 | N-(2-amino-6-chloro-pyridin-3-ylmet...)
Affinity DataEC50:  8nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230591(3-(acetylthio)-4-(N-((2-amino-6-methylpyridin-3-yl...)
Affinity DataEC50:  8nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230592(CHEMBL251889 | N-(2-amino-pyridin-3-ylmethyl)-N-{2...)
Affinity DataEC50:  479nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230593(3-(2-amino-6-chloro-pyridin-3-ylmethyl)-5-(2-hydro...)
Affinity DataEC50:  9nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230595(CHEMBL251888 | N-{2-[2-[acetyl-(2-amino-6-methyl-p...)
Affinity DataEC50:  32nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230594((4-(N-((2-amino-6-methylpyridin-3-yl)methyl)formam...)
Affinity DataEC50:  116nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230596(3-(2-amino-6-methyl-pyridin-3-ylmethyl)-5-(2-hydro...)
Affinity DataEC50:  9.54E+3nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230597(4-(N-((2-amino-6-methylpyridin-3-yl)methyl)formami...)
Affinity DataEC50:  28nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230598(CHEMBL253045 | N-((2-amino-6-methylpyridin-3-yl)me...)
Affinity DataEC50:  13nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230599(3-(2-(4-(N-((2-amino-6-methylpyridin-3-yl)methyl)f...)
Affinity DataEC50:  52nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230600(3-(2-amino-6-methyl-pyridin-3-ylmethyl)-5-(2-hydro...)
Affinity DataEC50:  18nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230601(CHEMBL401964 | N-((2-amino-6-methylpyridin-3-yl)me...)
Affinity DataEC50:  6.00E+3nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransketolase(Homo sapiens (Human))
Array Biopharma

Curated by ChEMBL
LigandPNGBDBM50230587(CHEMBL440237 | N-(2-amino-6-methyl-pyridin-3-ylmet...)
Affinity DataEC50:  12nMAssay Description:Inhibition of transketolase in human HCT116 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed