Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with all data for entry = 50038098
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371414(CHEMBL271828)
Affinity DataIC50:  0.5nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50233341(2-(3-isopropylureido)-N-(2-((1S,2R)-2-(4-(methylth...)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371414(CHEMBL271828)
Affinity DataIC50:  3.70nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371413(CHEMBL270959)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50233341(2-(3-isopropylureido)-N-(2-((1S,2R)-2-(4-(methylth...)
Affinity DataIC50:  5.10nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50233341(2-(3-isopropylureido)-N-(2-((1S,2R)-2-(4-(methylth...)
Affinity DataIC50:  7.5nMAssay Description:Binding affinity to wild type CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371414(CHEMBL271828)
Affinity DataIC50:  9nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50233341(2-(3-isopropylureido)-N-(2-((1S,2R)-2-(4-(methylth...)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371423(CHEMBL270906)
Affinity DataIC50:  21nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371413(CHEMBL270959)
Affinity DataIC50:  23nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371412(CHEMBL411726)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371412(CHEMBL411726)
Affinity DataIC50:  37nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371423(CHEMBL270906)
Affinity DataIC50:  42nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371413(CHEMBL270959)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371415(CHEMBL272168)
Affinity DataIC50:  64nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371424(CHEMBL429425)
Affinity DataIC50:  87nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371423(CHEMBL270906)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371412(CHEMBL411726)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371415(CHEMBL272168)
Affinity DataIC50:  215nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of MCP1-induced calcium fluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371416(CHEMBL273079)
Affinity DataIC50:  268nMAssay Description:Binding affinity to wild type CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371427(CHEMBL271537)
Affinity DataIC50:  360nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371428(CHEMBL271752)
Affinity DataIC50:  400nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371429(CHEMBL270957)
Affinity DataIC50:  530nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371422(CHEMBL269898)
Affinity DataIC50:  540nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371425(CHEMBL411935)
Affinity DataIC50:  550nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371416(CHEMBL273079)
Affinity DataIC50:  790nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371419(CHEMBL408172)
Affinity DataIC50:  970nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371421(CHEMBL409712)
Affinity DataIC50:  1.19E+3nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371415(CHEMBL272168)
Affinity DataIC50:  1.20E+3nMAssay Description:Antagonist activity at human CCR2 in PBMCs assessed as inhibition of chemotaxisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371417(CHEMBL406925)
Affinity DataIC50:  2.17E+3nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371430(CHEMBL272860)
Affinity DataIC50:  3.01E+3nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371426(CHEMBL272167)
Affinity DataIC50:  4.13E+3nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371426(CHEMBL272167)
Affinity DataIC50:  4.13E+3nMAssay Description:Binding affinity to wild type CCR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371420(CHEMBL272407)
Affinity DataIC50:  7.86E+3nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371418(CHEMBL407145)
Affinity DataIC50:  1.20E+4nMAssay Description:Displacement of radiolabeled MCP1 from human CCR2 in PBMCsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed