Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50025806
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266500(CHEMBL515991 | Methyl 7-(2-(2-(biphenyl-4-yl)-5-me...)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266531(CHEMBL458648 | Methyl 7-(2-(2-(4-methoxyphenyl)-5-...)
Affinity DataEC50:  5.25E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266532(CHEMBL458866 | Methyl 7-(2-(2-(4-methoxyphenyl)-5-...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266533(CHEMBL458867 | Methyl 7-(2-(2-(3-methoxyphenyl)-5-...)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266534(CHEMBL514441 | Methyl 7-(2-(2-(3-methoxyphenyl)-5-...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266548(CHEMBL458221 | Methyl 7-(2-(2-(4-tert-butylphenyl)...)
Affinity DataEC50:  2.29E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266549(CHEMBL514568 | Methyl 7-(2-(2-(4-tert-butylphenyl)...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266550(CHEMBL456912 | Methyl 7-(2-(5-methyl-2-p-tolyloxaz...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266551(CHEMBL515666 | Methyl 7-(2-(5-methyl-2-p-tolyloxaz...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266569(CHEMBL475988 | Methyl 7-(2-(5-methyl-2-m-tolyloxaz...)
Affinity DataEC50:  1.55E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266570(CHEMBL475989 | Methyl 7-(2-(5-methyl-2-(3-(trifluo...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266571(CHEMBL476197 | Methyl 7-(2-(5-methyl-2-(3-(trifluo...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266595(CHEMBL514713 | Methyl 7-(2-(2-(4-fluorophenyl)-5-m...)
Affinity DataEC50:  70nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266596(CHEMBL443910 | Methyl 7-(2-(2-(4-fluorophenyl)-5-m...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266597(CHEMBL514381 | Methyl 7-(2-(2-(3-fluorophenyl)-5-m...)
Affinity DataEC50:  1.29E+3nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266598(CHEMBL477644 | Methyl 7-(2-(2-(3-fluorophenyl)-5-m...)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50240768(7-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-2-oxo...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM24566(2-({4-chloro-6-[(2,3-dimethylphenyl)amino]pyrimidi...)
Affinity DataEC50:  1.20E+4nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266500(CHEMBL515991 | Methyl 7-(2-(2-(biphenyl-4-yl)-5-me...)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266501(CHEMBL455853 | Methyl 7-(2-(2-(biphenyl-4-yl)-5-me...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266531(CHEMBL458648 | Methyl 7-(2-(2-(4-methoxyphenyl)-5-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266532(CHEMBL458866 | Methyl 7-(2-(2-(4-methoxyphenyl)-5-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266533(CHEMBL458867 | Methyl 7-(2-(2-(3-methoxyphenyl)-5-...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266534(CHEMBL514441 | Methyl 7-(2-(2-(3-methoxyphenyl)-5-...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266548(CHEMBL458221 | Methyl 7-(2-(2-(4-tert-butylphenyl)...)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266549(CHEMBL514568 | Methyl 7-(2-(2-(4-tert-butylphenyl)...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266550(CHEMBL456912 | Methyl 7-(2-(5-methyl-2-p-tolyloxaz...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266551(CHEMBL515666 | Methyl 7-(2-(5-methyl-2-p-tolyloxaz...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266568(CHEMBL515454 | Methyl 7-(2-(5-methyl-2-m-tolyloxaz...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266569(CHEMBL475988 | Methyl 7-(2-(5-methyl-2-m-tolyloxaz...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266570(CHEMBL475989 | Methyl 7-(2-(5-methyl-2-(3-(trifluo...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266571(CHEMBL476197 | Methyl 7-(2-(5-methyl-2-(3-(trifluo...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266595(CHEMBL514713 | Methyl 7-(2-(2-(4-fluorophenyl)-5-m...)
Affinity DataEC50:  1.62E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266596(CHEMBL443910 | Methyl 7-(2-(2-(4-fluorophenyl)-5-m...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266597(CHEMBL514381 | Methyl 7-(2-(2-(3-fluorophenyl)-5-m...)
Affinity DataEC50:  960nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266598(CHEMBL477644 | Methyl 7-(2-(2-(3-fluorophenyl)-5-m...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266609(CHEMBL478897 | Methyl 7-(2-(5-methyl-2-(3-nitrophe...)
Affinity DataEC50:  3.55E+3nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50240768(7-[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethoxy]-2-oxo...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARgamma in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50266501(CHEMBL455853 | Methyl 7-(2-(2-(biphenyl-4-yl)-5-me...)
Affinity DataEC50:  910nMAssay Description:Agonist activity at human PPARalpha in U2OS cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed