Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50038346
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375279(CHEMBL270181)
Affinity DataIC50:  0.580nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375280(CHEMBL404189)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375286(CHEMBL256193)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375267(CHEMBL410195)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375278(CHEMBL256192)
Affinity DataIC50:  0.980nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375281(CHEMBL270417)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375273(CHEMBL255183)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375277(CHEMBL404152)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM91872(Chk1_152)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375270(CHEMBL257067)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375272(CHEMBL404479)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375285(CHEMBL257703)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375275(CHEMBL272347)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM91859(Chk1_136)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375271(CHEMBL272711)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375284(CHEMBL411098)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375268(CHEMBL257317)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50218722(3-(3-methoxy-4-nitro-phenyl)-5,10-dihydro-dibenzo[...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375282(CHEMBL271727)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375269(CHEMBL404498)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375274(CHEMBL427720)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375283(CHEMBL255816)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375276(CHEMBL404021)
Affinity DataIC50:  1.05E+3nMAssay Description:Inhibition of recombinant Chk1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM91859(Chk1_136)
Affinity DataEC50:  50nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375285(CHEMBL257703)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375280(CHEMBL404189)
Affinity DataEC50:  280nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375270(CHEMBL257067)
Affinity DataEC50:  900nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375267(CHEMBL410195)
Affinity DataEC50:  70nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375286(CHEMBL256193)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM91872(Chk1_152)
Affinity DataEC50:  40nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375283(CHEMBL255816)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375281(CHEMBL270417)
Affinity DataEC50:  220nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375271(CHEMBL272711)
Affinity DataEC50:  50nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375282(CHEMBL271727)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375275(CHEMBL272347)
Affinity DataEC50:  200nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375274(CHEMBL427720)
Affinity DataEC50:  2.10E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375277(CHEMBL404152)
Affinity DataEC50:  3.10E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375278(CHEMBL256192)
Affinity DataEC50:  2.60E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375272(CHEMBL404479)
Affinity DataEC50:  600nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375268(CHEMBL257317)
Affinity DataEC50:  350nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375269(CHEMBL404498)
Affinity DataEC50:  3.50E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375273(CHEMBL255183)
Affinity DataEC50:  1.50E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375284(CHEMBL411098)
Affinity DataEC50:  200nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50375279(CHEMBL270181)
Affinity DataEC50:  3.10E+3nMAssay Description:Inhibition of human Chk1 in H1299 cells assessed as blockade of Cdc25A degradationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed