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PubMed code 18394907

Compile data set for download or QSAR
Found 23 hits of Enzyme Inhibition Constant Data   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34017
PNG
(CHEMBL104850 | phenylpropanoic acid derivative, 7)
Show SMILES Cc1oc(nc1CCOc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C25H24N2O4/c1-18-22(26-24(31-18)20-7-3-2-4-8-20)13-16-30-21-11-9-19(10-12-21)17-23(25(28)29)27-14-5-6-15-27/h2-12,14-15,23H,13,16-17H2,1H3,(H,28,29)/t23-/m0/s1
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n/an/a 29n/a 26n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM33284
PNG
(BMC164883 Compound 53 | phenylpropanoic acid deriv...)
Show SMILES Cc1oc(nc1CCCc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C26H26N2O3/c1-19-23(27-25(31-19)22-9-3-2-4-10-22)11-7-8-20-12-14-21(15-13-20)18-24(26(29)30)28-16-5-6-17-28/h2-6,9-10,12-17,24H,7-8,11,18H2,1H3,(H,29,30)/t24-/m0/s1
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Article
PubMed
n/an/a 185n/a 140n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34025
PNG
(phenylpropanoic acid derivative, 40)
Show SMILES Cc1oc(nc1C\C=C\c1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C26H24N2O3/c1-19-23(27-25(31-19)22-9-3-2-4-10-22)11-7-8-20-12-14-21(15-13-20)18-24(26(29)30)28-16-5-6-17-28/h2-10,12-17,24H,11,18H2,1H3,(H,29,30)/b8-7+/t24-/m0/s1
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n/an/a 255n/a 102n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34018
PNG
(phenylpropanoic acid derivative, 28)
Show SMILES Cc1oc(nc1CC#Cc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C26H22N2O3/c1-19-23(27-25(31-19)22-9-3-2-4-10-22)11-7-8-20-12-14-21(15-13-20)18-24(26(29)30)28-16-5-6-17-28/h2-6,9-10,12-17,24H,11,18H2,1H3,(H,29,30)/t24-/m0/s1
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n/an/a 293n/a 173n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34030
PNG
(phenylpropanoic acid derivative, 56 | racemic)
Show SMILES Cc1oc(nc1CCCc1ccc(CC(C(O)=O)c2ccc(cc2)-c2ccccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C34H31NO3/c1-24-32(35-33(38-24)30-12-6-3-7-13-30)14-8-9-25-15-17-26(18-16-25)23-31(34(36)37)29-21-19-28(20-22-29)27-10-4-2-5-11-27/h2-7,10-13,15-22,31H,8-9,14,23H2,1H3,(H,36,37)
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n/an/a 587n/a 1.80E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34034
PNG
(phenylpropanoic acid derivative, 66)
Show SMILES Cc1oc(nc1CCNc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C25H25N3O3/c1-18-22(27-24(31-18)20-7-3-2-4-8-20)13-14-26-21-11-9-19(10-12-21)17-23(25(29)30)28-15-5-6-16-28/h2-12,15-16,23,26H,13-14,17H2,1H3,(H,29,30)/t23-/m0/s1
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n/an/a 1.60E+3n/a 480n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34027
PNG
(phenylpropanoic acid derivative, 44)
Show SMILES CN(C\C=C\c1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)c1ccccc1
Show InChI InChI=1S/C23H24N2O2/c1-24(21-9-3-2-4-10-21)15-7-8-19-11-13-20(14-12-19)18-22(23(26)27)25-16-5-6-17-25/h2-14,16-17,22H,15,18H2,1H3,(H,26,27)/b8-7+/t22-/m0/s1
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n/an/a 2.00E+3n/a 3.70E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34020
PNG
(phenylpropanoic acid derivative, 30 | racemic)
Show SMILES Cc1oc(nc1CC#Cc1ccc(CC(C(O)=O)c2ccc(cc2)-c2ccccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C34H27NO3/c1-24-32(35-33(38-24)30-12-6-3-7-13-30)14-8-9-25-15-17-26(18-16-25)23-31(34(36)37)29-21-19-28(20-22-29)27-10-4-2-5-11-27/h2-7,10-13,15-22,31H,14,23H2,1H3,(H,36,37)
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n/an/a 2.20E+3n/a 2.50E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34026
PNG
(phenylpropanoic acid derivative, 41)
Show SMILES Cc1oc(nc1C\C=C\c1ccc(C[C@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C26H24N2O3/c1-19-23(27-25(31-19)22-9-3-2-4-10-22)11-7-8-20-12-14-21(15-13-20)18-24(26(29)30)28-16-5-6-17-28/h2-10,12-17,24H,11,18H2,1H3,(H,29,30)/b8-7+/t24-/m1/s1
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n/an/a 2.60E+3n/a 2.60E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34031
PNG
(phenylpropanoic acid derivative, 57 | racemic)
Show SMILES Cc1oc(nc1CCCc1ccc(CC(C(O)=O)c2cccc(c2)-c2ccccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C34H31NO3/c1-24-32(35-33(38-24)28-13-6-3-7-14-28)17-8-10-25-18-20-26(21-19-25)22-31(34(36)37)30-16-9-15-29(23-30)27-11-4-2-5-12-27/h2-7,9,11-16,18-21,23,31H,8,10,17,22H2,1H3,(H,36,37)
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n/an/a 2.80E+3n/a 4.00E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34021
PNG
(phenylpropanoic acid derivative, 31 | racemic)
Show SMILES Cc1oc(nc1CC#Cc1ccc(CC(C(O)=O)c2cccc(c2)-c2ccccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C34H27NO3/c1-24-32(35-33(38-24)28-13-6-3-7-14-28)17-8-10-25-18-20-26(21-19-25)22-31(34(36)37)30-16-9-15-29(23-30)27-11-4-2-5-12-27/h2-7,9,11-16,18-21,23,31H,17,22H2,1H3,(H,36,37)
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n/an/a 2.80E+3n/a 1.30E+4n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34028
PNG
(phenylpropanoic acid derivative, 54)
Show SMILES Cc1oc(nc1CCCc1ccc(C[C@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C26H26N2O3/c1-19-23(27-25(31-19)22-9-3-2-4-10-22)11-7-8-20-12-14-21(15-13-20)18-24(26(29)30)28-16-5-6-17-28/h2-6,9-10,12-17,24H,7-8,11,18H2,1H3,(H,29,30)/t24-/m1/s1
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n/an/a 3.10E+3n/a 2.30E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM33296
PNG
(BMC164883 Compound 58 | phenylpropanoic acid deriv...)
Show SMILES Cc1oc(nc1CCCc1ccc(CC(C(O)=O)c2ccccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C28H27NO3/c1-20-26(29-27(32-20)24-12-6-3-7-13-24)14-8-9-21-15-17-22(18-16-21)19-25(28(30)31)23-10-4-2-5-11-23/h2-7,10-13,15-18,25H,8-9,14,19H2,1H3,(H,30,31)
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n/an/a 4.00E+3n/a 3.90E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34033
PNG
(phenylpropanoic acid derivative, 60)
Show SMILES CN(CCCc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)c1ccccc1
Show InChI InChI=1S/C23H26N2O2/c1-24(21-9-3-2-4-10-21)15-7-8-19-11-13-20(14-12-19)18-22(23(26)27)25-16-5-6-17-25/h2-6,9-14,16-17,22H,7-8,15,18H2,1H3,(H,26,27)/t22-/m0/s1
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n/an/a 1.10E+4n/a 3.60E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34024
PNG
(phenylpropanoic acid derivative, 36)
Show SMILES CN(C\C=C\c1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)c1ccccn1
Show InChI InChI=1S/C22H23N3O2/c1-24(21-8-2-3-13-23-21)14-6-7-18-9-11-19(12-10-18)17-20(22(26)27)25-15-4-5-16-25/h2-13,15-16,20H,14,17H2,1H3,(H,26,27)/b7-6+/t20-/m0/s1
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n/an/a 1.20E+4n/a 492n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34023
PNG
(phenylpropanoic acid derivative, 33)
Show SMILES CN(CC#Cc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)c1ccccc1
Show InChI InChI=1S/C23H22N2O2/c1-24(21-9-3-2-4-10-21)15-7-8-19-11-13-20(14-12-19)18-22(23(26)27)25-16-5-6-17-25/h2-6,9-14,16-17,22H,15,18H2,1H3,(H,26,27)/t22-/m0/s1
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n/an/a 1.20E+4n/a 2.00E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34029
PNG
(phenylpropanoic acid derivative, 55 | racemic)
Show SMILES Cc1oc(nc1CCCc1ccc(CC(C(O)=O)c2cccnc2)cc1)-c1ccccc1
Show InChI InChI=1S/C27H26N2O3/c1-19-25(29-26(32-19)22-8-3-2-4-9-22)11-5-7-20-12-14-21(15-13-20)17-24(27(30)31)23-10-6-16-28-18-23/h2-4,6,8-10,12-16,18,24H,5,7,11,17H2,1H3,(H,30,31)
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n/an/a 2.20E+4n/a 3.90E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34019
PNG
(phenylpropanoic acid derivative, 29 | racemic)
Show SMILES Cc1oc(nc1CC#Cc1ccc(CC(C(O)=O)c2cccnc2)cc1)-c1ccccc1
Show InChI InChI=1S/C27H22N2O3/c1-19-25(29-26(32-19)22-8-3-2-4-9-22)11-5-7-20-12-14-21(15-13-20)17-24(27(30)31)23-10-6-16-28-18-23/h2-4,6,8-10,12-16,18,24H,11,17H2,1H3,(H,30,31)
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n/an/a 2.60E+4n/a 4.50E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34032
PNG
(phenylpropanoic acid derivative, 59)
Show SMILES CN(CCCc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)c1ccccn1
Show InChI InChI=1S/C22H25N3O2/c1-24(21-8-2-3-13-23-21)14-6-7-18-9-11-19(12-10-18)17-20(22(26)27)25-15-4-5-16-25/h2-5,8-13,15-16,20H,6-7,14,17H2,1H3,(H,26,27)/t20-/m0/s1
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n/an/a 2.80E+4n/a 1.20E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34035
PNG
(phenylpropanoic acid derivative, 74)
Show SMILES Cc1oc(nc1CNCc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1)-c1ccccc1
Show InChI InChI=1S/C25H25N3O3/c1-18-22(27-24(31-18)21-7-3-2-4-8-21)17-26-16-20-11-9-19(10-12-20)15-23(25(29)30)28-13-5-6-14-28/h2-14,23,26H,15-17H2,1H3,(H,29,30)/t23-/m0/s1
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n/an/a>5.00E+4n/a 9.00E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34022
PNG
(phenylpropanoic acid derivative, 32 | racemic)
Show SMILES CN(CC#Cc1ccc(CC(C(O)=O)n2cccc2)cc1)c1ccccn1
Show InChI InChI=1S/C22H21N3O2/c1-24(21-8-2-3-13-23-21)14-6-7-18-9-11-19(12-10-18)17-20(22(26)27)25-15-4-5-16-25/h2-5,8-13,15-16,20H,14,17H2,1H3,(H,26,27)
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n/an/a 5.30E+4n/a 9.00E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34037
PNG
(phenylpropanoic acid derivative, 76)
Show SMILES CC(=O)N(Cc1nc(oc1C)-c1ccccc1)Cc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1
Show InChI InChI=1S/C27H27N3O4/c1-19-24(28-26(34-19)23-8-4-3-5-9-23)18-30(20(2)31)17-22-12-10-21(11-13-22)16-25(27(32)33)29-14-6-7-15-29/h3-15,25H,16-18H2,1-2H3,(H,32,33)/t25-/m0/s1
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n/an/a>1.00E+5n/a>3.00E+4n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
Peroxisome proliferator-activated receptor


(Homo sapiens (Human))
BDBM34036
PNG
(phenylpropanoic acid derivative, 75)
Show SMILES CN(Cc1nc(oc1C)-c1ccccc1)Cc1ccc(C[C@@H](C(O)=O)n2cccc2)cc1
Show InChI InChI=1S/C26H27N3O3/c1-19-23(27-25(32-19)22-8-4-3-5-9-22)18-28(2)17-21-12-10-20(11-13-21)16-24(26(30)31)29-14-6-7-15-29/h3-15,24H,16-18H2,1-2H3,(H,30,31)/t24-/m0/s1
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n/an/a>1.00E+5n/a 7.00E+3n/an/a7.423



Pfizer Inc



Assay Description
Human 6His-PPAR gamma ligand-binding domain was added to the mixture containing radioligand and test compound, followed by yttrium silicate polylysin...


Bioorg Med Chem 16: 4883-907 (2008)


Article DOI: 10.1016/j.bmc.2008.03.043
BindingDB Entry DOI: 10.7270/Q2SN0797
More data for this
Ligand-Target Pair
* indicates data uncertainty>20%