Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50038861
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50073850((S)-2-((S)-2-Benzyloxycarbonylamino-3-methyl-butyr...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249628((S)-N-(4-amino-3,4-dioxo-1-phenylbutan-2-yl)-3-met...)
Affinity DataIC50:  2.81E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249635((S)-N-(4-(4-methoxyphenethylamino)-3,4-dioxo-1-phe...)
Affinity DataIC50:  6.19E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249620((S)-N-(4-(4-methoxybenzylamino)-3,4-dioxo-1-phenyl...)
Affinity DataIC50:  6.19E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249634((S)-N-(3,4-dioxo-4-(phenethylamino)-1-phenylbutan-...)
Affinity DataIC50:  7.41E+3nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249632((S)-N-(4-(4-fluorobenzylamino)-3,4-dioxo-1-phenylb...)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249622((S)-N-(3,4-dioxo-1-phenyl-4-(2-(pyridin-2-yl)ethyl...)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249621((S)-N-(4-(3,4-dimethoxybenzylamino)-3,4-dioxo-1-ph...)
Affinity DataIC50:  3.53E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249630((S)-N-(4-(ethylamino)-3,4-dioxo-1-phenylbutan-2-yl...)
Affinity DataIC50:  4.02E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249619((S)-N-(4-(benzylamino)-3,4-dioxo-1-phenylbutan-2-y...)
Affinity DataIC50:  6.46E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249633((S)-N-(3,4-dioxo-1-phenyl-4-(pyridin-2-ylmethylami...)
Affinity DataIC50:  8.48E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249629((S)-3-methyl-N-(4-(methylamino)-3,4-dioxo-1-phenyl...)
Affinity DataIC50:  9.14E+4nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCalpain-1 catalytic subunit(Homo sapiens (Human))
Kyung Hee University

Curated by ChEMBL
LigandPNGBDBM50249631((S)-N-(4-(isopropylamino)-3,4-dioxo-1-phenylbutan-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human erythrocytes mu-calpain by spectrofluorimeterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed