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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM24182 (4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet  | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 420 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair |  3D Structure (crystal) | ||||||||||||
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM50009131 (4-Amino-3-(2,4-dichloro-phenyl)-butyric acid; hydr...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM50009136 ((7-Aminomethyl-bicyclo[4.2.0]octa-1(6),2,4-trien-7...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM50009132 ((1-Aminomethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM50009134 ((1-Aminomethyl-indan-1-yl)-acetic acid; hydrochlor...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM50009133 (4-Amino-3-(2,6-dichloro-phenyl)-butyric acid; hydr...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| GABA-B receptor 1/2 (Rattus norvegicus) | BDBM50009135 ((1-Aminomethyl-5-chloro-indan-1-yl)-acetic acid; h...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Neurochimie du CNRS Curated by ChEMBL | Assay Description Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptor | Citation and Details | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
