Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50035946
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)
Affinity DataIC50:  420nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50009131(4-Amino-3-(2,4-dichloro-phenyl)-butyric acid; hydr...)
Affinity DataIC50:  1.10E+4nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50009132((1-Aminomethyl-1,2,3,4-tetrahydro-naphthalen-1-yl)...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50009134((1-Aminomethyl-indan-1-yl)-acetic acid; hydrochlor...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50009133(4-Amino-3-(2,6-dichloro-phenyl)-butyric acid; hydr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50009135((1-Aminomethyl-5-chloro-indan-1-yl)-acetic acid; h...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid type B receptor subunit 1/2(Rattus norvegicus (Rat))
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50009136((7-Aminomethyl-bicyclo[4.2.0]octa-1(6),2,4-trien-7...)
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of [3H]baclofen from gamma-aminobutyric-acid B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed